Patent International Class: C07D 413/6

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Indole compounds bearing aryl or heteroaryl groups having sphingosine-1-phosphate (S1P) receptor biological activity
Inventor: Beard, et al. | Patent Number: 8143291

Heterocyclyl compounds
Inventor: Adam, et al. | Patent Number: 8138175

Long wavelength thiol-reactive fluorophores
Inventor: Pitner, et al. | Patent Number: 8129525

Antifungal compounds containing benzothiazinone, benzoxazinone or benzoxazolinone and process thereof
Inventor: Borate, et al. | Patent Number: 8129369

Compounds and compositions as protein kinase inhibitors
Inventor: Wan, et al. | Patent Number: 8101608

Cycloalkyl derivatives of 3-hydroxy-4-pyridinones
Inventor: Tam, et al. | Patent Number: 8097624

Substituted spirochromanone derivatives
Inventor: Iino, et al. | Patent Number: 8093389

HIV inhibiting pyrimidines derivatives
Inventor: Guillemont, et al. | Patent Number: 8080551

Long wavelength thiol-reactive fluorophores
Inventor: Pitner, et al. | Patent Number: 8071794

Phenolic and catecholic amines and prodrugs thereof
Inventor: Puschl, et al. | Patent Number: 8067410

Chemical compounds
Inventor: Turnbull, et al. | Patent Number: 8026262

Compounds with antiparasitic activity and medicines containing same
Inventor: Vial, et al. | Patent Number: 8012985

Derivatives of 1-{[1,5-bis(4-chlorophenyl)-2-methyl-1H-pyrrol-3-yl]methyl}-4-methylpiper- azine, synthesis process and uses thereof
Inventor: Biava, et al. | Patent Number: 8012970

Functionalized diarylisoxazoles inhibitors of ciclooxygenase
Inventor: Scilimati, et al. | Patent Number: 7989450

ALPHA2C adrenoreceptor agonists
Inventor: McCormick, et al. | Patent Number: 7985748

Substituted isoxazoles as fungicides
Inventor: Lee, et al. | Patent Number: 7977341

Indolone-acetamide derivatives, processes for preparing them and their uses
Inventor: Starck, et al. | Patent Number: 7964593

Useful indole compounds
Inventor: Bartolini, et al. | Patent Number: 7960544

Substituted gamma lactams as therapeutic agents
Inventor: Old, et al. | Patent Number: 7960381

Piperidine compounds for use as orexin receptor antagonist
Inventor: Chan, et al. | Patent Number: 7943645

Heterocyclic amide compounds useful as kinase inhibitors
Inventor: Wrobleski, et al. | Patent Number: 7935696

Chiral bisoxazoline catalysts
Inventor: Ying, et al. | Patent Number: 7919422

Process for {3-[2(R)-[(1R)-1-[3,5-bis(trifluoromethyl)phenyl]ethoxy]-3(S)-(4-fluoroph- enyl)morpholin-4-yl]methyl]-5-oxo-4,5-dihydro-[1,2,4]-triazol-1-yl}phospho- nic acid
Inventor: McNamara, et al. | Patent Number: 7915407

Indole compounds bearing aryl or heteroaryl groups having sphingosine 1-phosphate (S1P) receptor biological activity
Inventor: Beard, et al. | Patent Number: 7888336

Substituted gamma lactams as therapeutic agents
Inventor: Old, et al. | Patent Number: 7879854

Oxindole derivative as feeding control agent
Inventor: Tokunaga, et al. | Patent Number: 7825155

Aminomethyl beta-secretase inhibitors for the treatment of alzheimer's disease
Inventor: Coburn, et al. | Patent Number: 7820674

Cyclized derivatives as Eg-5 inhibitors
Inventor: Boyce, et al. | Patent Number: 7820646

Brain/neuronal cell-protecting agent and therapeutic agent for sleep disorder
Inventor: Matsumoto, et al. | Patent Number: 7812025

Process for {3-[2(R)-[(1R)-1-[3,5-bis(trifluoromethyl) phenyl]ethoxy]-3(S)-(4-fluorophenyl)morpholin-4-yl]methyl]-5-oxo-4,5-dihy- dro-[1,2,4]-triazol-1-yl}phosphonic acid
Inventor: McNamara, et al. | Patent Number: 7807829

Substituted pyrimidinones
Inventor: Durley | Patent Number: 7795271

Monocyclic and bicyclic compounds and methods of use
Inventor: Zhang, et al. | Patent Number: 7790726

Benzimidazole derivatives: preparation and pharmaceutical applications
Inventor: Chen, et al. | Patent Number: 7781595

Thienopyrroles as antiviral agents
Inventor: Attenni, et al. | Patent Number: 7781431

Substituted thieno[3,2-d]pyridines as inhibitors of the VEGF receptor and HGF receptor
Inventor: Vaisburg, et al. | Patent Number: 7772247

Long wavelength thiol-reactive fluorophores
Inventor: Pitner, et al. | Patent Number: 7767821

Substituted piperidine derivatives as somatostatin SST1 receptor antagonists
Inventor: Hoyer, et al. | Patent Number: 7754719

Cyanine compounds, optical filters, and optical recording materials
Inventor: Aoyama, et al. | Patent Number: 7745632

Tetrahydronaphthyridine and tetrahydropyrido[4,3-d]pyrimidine compounds and compositions thereof useful in the treatment of conditions associated with neurological and inflammatory disorders and dysfunctions
Inventor: Kelly, et al. | Patent Number: 7745451

Antifungal bicyclic hetero ring compounds
Inventor: Kawakami, et al. | Patent Number: 7737166

Process for making heteroaryl amine intermediate compounds
Inventor: Li, et al. | Patent Number: 7714127

Fused heteroaryl derivatives for use as p38 kinase inhibitors in the treatment of I.A. rheumatoid arthritis
Inventor: Campos, et al. | Patent Number: 7687532

Cyclopropyl amines as modulators of the histamine H.sub.3 receptor
Inventor: Allison, et al. | Patent Number: 7687499

2-amino-7,8-dihydro-6H-pyrido[4,3-d]pyrimidin-5-ones
Inventor: Machajewski, et al. | Patent Number: 7671059

Herbicide combination
Inventor: Hills, et al. | Patent Number: 7648945

Benzimidazole derivatives
Inventor: Frenkel, et al. | Patent Number: 7635774

Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
Inventor: Barf, et al. | Patent Number: 7618961

Substituted pyrazolo[1,5-a]pyrimidines as protein kinase inhibitors
Inventor: Guzi, et al. | Patent Number: 7605155

Aryl sulfamide derivatives and methods of their use
Inventor: McComas, et al. | Patent Number: 7601722

Morpholinyl piperidine glycine transporter inhibitors
Inventor: Lindsley, et al. | Patent Number: 7576083

Chemical compounds
Inventor: Turnbull, et al. | Patent Number: 7572820

1,3,4-Substituted pyrazoles as 5-HT receptor antagonists for the treatment of psychoses and neurological disorders
Inventor: Schiemann, et al. | Patent Number: 7566709

Long wavelength thiol-reactive fluorophores
Inventor: Pitner, et al. | Patent Number: 7563891

Substituted Imidazo[1,2-a]pyridines as Antibacterial Agents
Inventor: Sciotti, et al. | Patent Number: 7563788

Herbicide-safener combination
Inventor: Hills, et al. | Patent Number: 7563749

Indoles are cannabinoid receptor ligands
Inventor: Frost, et al. | Patent Number: 7560481

Use of sulfonylureas
Inventor: Hills, et al. | Patent Number: 7557066

Piperazinediones as oxytocin receptor antagonists
Inventor: Borthwick, et al. | Patent Number: 7550462

Aryl-4-ethynyl-isoxazole derivatives
Inventor: Buettelmann, et al. | Patent Number: 7544704

N-substituted piperidine derivatives as serotonin receptor agents
Inventor: Andersson, et al. | Patent Number: 7538222

Substituted pyrrolo[3,2-d]pyrimidines as glycogen synthase kinase (GSK) inhibitors
Inventor: Kataoka, et al. | Patent Number: 7528140

4-arylmorpholin-3-one derivatives, their preparation and therapeutic use thereof
Inventor: Emonds-Alt, et al. | Patent Number: 7521449

Heterocyclic inhibitors of MEK and methods of use thereof
Inventor: Marlow, et al. | Patent Number: 7517994

Derivatives of sulphonamides, their preparation and use as medicaments
Inventor: Merce-Vidal, et al. | Patent Number: 7498328

Pyrrolidinyl beta-amino amide-based inhibitors of dipeptidyl peptidase IV and methods
Inventor: O'Connor, et al. | Patent Number: 7488725

HIV integrase inhibitors
Inventor: Wai, et al. | Patent Number: 7476666

Azole methylidene cyanide derivatives and their use as protein kinase modulators
Inventor: Gaillard, et al. | Patent Number: 7465736

Substituted pyrrolo[2.3-B]pyridines
Inventor: Ahmed, et al. | Patent Number: 7465726

Acetylenyl-pyrazolo-pyrimidine derivatives
Inventor: Gatti McArthur, et al. | Patent Number: 7446113

1H-pyrrolo [2,3-D] pyrimidine derivatives and methods of use thereof
Inventor: Tanaka, et al. | Patent Number: 7429596

Pyrrolidine derivatives as factor Xa inhibitors
Inventor: Chan, et al. | Patent Number: 7429587

Furo[2.3-b]pyridine derivatives for the treatment of hyper-proliferative disorders
Inventor: Zhang, et al. | Patent Number: 7429584

Compounds for treating fundic disaccomodation
Inventor: Van Emelen, et al. | Patent Number: 7423048

Stable crystalline form of bifeprunox mesylate, dosage forms thereof and methods for using same
Inventor: Eijgendaal, et al. | Patent Number: 7423040

Morpholine derivatives as norepinephrine reuptake inhibitors
Inventor: Campbell, et al. | Patent Number: 7423037

Gamma lactams as prostaglandin agonists and use thereof
Inventor: Araldi, et al. | Patent Number: 7419999

Stable crystalline form of bifeprunox mesylate (7-[4-([1,1'-biphenyl]-3-ylmethyl)-1-piperazinyl]-2(3H)-benzoxazolone monomethanesulfonate)
Inventor: Eijgendaal, et al. | Patent Number: 7405216

Substituted thienopyrimidinones as a mitotic kinesin inhibitor
Inventor: Fraley, et al. | Patent Number: 7378411

PNA monomer and precursor
Inventor: Kim, et al. | Patent Number: 7371860

Substituted aryl acylthioureas and related compounds; inhibitors of viral replication
Inventor: Phadke, et al. | Patent Number: 7365068

Non-peptide GnRH antagonists
Inventor: Roe, et al. | Patent Number: 7365065

Substituted oxadiazolidinediones
Inventor: Elokdah, et al. | Patent Number: 7351726

Substituted isoxazoles as fungicides
Inventor: Lee, et al. | Patent Number: 7338967

Mycobacterial inhibitors
Inventor: Guillemont, et al. | Patent Number: 7338949

Derivatives of N-[heteroaryl(piperidine-2-yl) methyl]benzamide, preparation method thereof and application of same in therapeutics
Inventor: Dargazanli, et al. | Patent Number: 7335670

Isochroman compounds for treatment of CNS disorders
Inventor: Agejas-Chicharro, et al. | Patent Number: 7335660

4-Amino-5-phenyl-7-cyclobutyl-pyrrolo(2,3-d)pyrimidine derivatives
Inventor: Capraro, et al. | Patent Number: 7326699

Peroxisome proliferator activated receptor alpha agonists
Inventor: Dominianni, et al. | Patent Number: 7304062

Inhibitors of cathepsin S
Inventor: Liu, et al. | Patent Number: 7297714

Oxazolo-and furopyrimidines and their use in medicaments against tumors
Inventor: Bold, et al. | Patent Number: 7294633

Phenylalkynes
Inventor: Apodaca, et al. | Patent Number: 7288540

Fluorinated di-aryl urea compounds
Inventor: Cirillo, et al. | Patent Number: 7279475

Method of synthesis of azole-containing amino acids
Inventor: Hlasta, et al. | Patent Number: 7259263

Dipeptidyl peptidase inhibitors for the treatment of diabetes
Inventor: Brockunier, et al. | Patent Number: 7253172

Substituted furopyrimidinones as a mitotic kinesin inhibitors
Inventor: Fraley, et al. | Patent Number: 7244723

Synthesis of indole thiazole compounds as ligands for the Ah receptor
Inventor: DeLuca, et al. | Patent Number: 7241900

Piperidine derivatives and their use as modulators of chemokine (especially CCR3) activity
Inventor: Sanganee, et al. | Patent Number: 7238691

Thiadiazole-amine compounds for the treatment of neurodegenerative disorders
Inventor: Chen | Patent Number: 7232820

Substituted 5-aminomethyl-1H-pyrrole-2-carboxamides
Inventor: Merla, et al. | Patent Number: 7229991

Heterocyclymethylpiperidines and -piperazines possessing affinity at 5ht-1 type receptors
Inventor: Ward | Patent Number: 7214674

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