Patent International Class: C07D 211/14

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Sulfonamides as TRPM8 modulators
Inventor: Macielag, et al. | Patent Number: 8148422

Piperidine derivatives and cosmetic compositions thereof
Inventor: Cavezza, et al. | Patent Number: 8129409

Histamine H3-receptor ligands and their therapeutic applications
Inventor: Bertrand, et al. | Patent Number: 8076329

Bridged ring structures as pharmaceutical agents
Inventor: Flatt, et al. | Patent Number: 7863298

Process for production of piperidine derivatives
Inventor: D'Ambra, et al. | Patent Number: 7678915

N-sulfonylcarboximidamide apoptosis promoters
Inventor: Elmore, et al. | Patent Number: 7585858

Methods for synthesis of prodrugs from 1-acyl-alkyl derivatives and compositions thereof
Inventor: Gallop, et al. | Patent Number: 7560483

N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
Inventor: Ko, et al. | Patent Number: 7550486

Piperidine derivatives useful as modulators of chemokine receptor activity
Inventor: Sanganee, et al. | Patent Number: 7482363

Amino substituted aryloxybenzylpiperidine derivatives
Inventor: Marzabadi, et al. | Patent Number: 7446204

Amide compounds having MCH-antagonistic activity and medicaments comprising these compounds
Inventor: Stenkamp, et al. | Patent Number: 7351719

Process for producing 1-benzyl-4-[(5,6-dimethoxy-1-indanon)-2-yl]methylpiperidine or hydrochloride thereof
Inventor: Imai | Patent Number: 7332606

Tricyclic aromatic and bis-phenyl sulfinyl derivatives
Inventor: Bacon, et al. | Patent Number: 7314875

Chemical compounds
Inventor: Sanganee, et al. | Patent Number: 7304077

1-alkyl-4-(3-substitutedphenyl)piperidines
Inventor: Wentland | Patent Number: 7265226

Derivatives of 3-phenyl-n-(2-(4-benzyl)-piperidin-1-yl)-ethyl)-acrylamid with ccr-3-receptor antagonistic activity for use in the treatment of inflammations and allergic conditions
Inventor: Bhalay, et al. | Patent Number: 7259173

Naphthaline derivatives as H3 inverse agonists
Inventor: McArthur, et al. | Patent Number: 7259158

Bicyclic inhibitors of hormone sensitive lipase
Inventor: Petry, et al. | Patent Number: 7208504

Polyarylcarboxamides useful as lipid lowering agents
Inventor: Meerpoel, et al. | Patent Number: 7169796

Benzosuberonylpiperdine compounds as analgesics
Inventor: Barlocco, et al. | Patent Number: 7115633

Substituted propargylamines
Inventor: Jakobi, et al. | Patent Number: 7084158

Gonadotropin-releasing hormone receptor antagonists and methods relating thereto
Inventor: Chen, et al. | Patent Number: 7081459

Process and intermediates for the preparation of 4-aryl piperidines
Inventor: Boice, et al. | Patent Number: 6998488

Process for production of piperidine derivatives
Inventor: D'Ambra, et al. | Patent Number: 6974872

Compounds
Inventor: Barlocco, et al. | Patent Number: 6969724

Processes for producing racemic piperidine derivative and for producing optically active piperidine derivative
Inventor: Fujino, et al. | Patent Number: 6962998

Calcium channel blockers comprising two benzhydril moieties
Inventor: Snutch, et al. | Patent Number: 6951862

Calcium channel blockers comprising two benzhydril moieties
Inventor: Snutch, et al. | Patent Number: 6949554

Calcium channel inhibitors comprising benzhydril spaced from piperazine
Inventor: Snutch, et al. | Patent Number: 6943168

Process for production of piperidine derivatives
Inventor: D'Ambra, et al. | Patent Number: 6919458

Process for production of piperidine derivatives
Inventor: D'Ambra, et al. | Patent Number: 6919458

N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
Inventor: Ko, et al. | Patent Number: 6919368

Substituted tetrahydroisoquinolines as C5a receptor modulators
Inventor: Lee, et al. | Patent Number: 6916830

Phenoxyalkylamine derivatives useful as opioid .delta. receptor agonists
Inventor: Tsushima, et al. | Patent Number: 6916822

N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
Inventor: Ko, et al. | Patent Number: 6906066

N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
Inventor: Ko, et al. | Patent Number: 6897234

Phenylalkynes
Inventor: Apodaca, et al. | Patent Number: 6884803

N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
Inventor: Ko, et al. | Patent Number: 6875776

Arylamines as inhibitors of chemokine binding to US28
Inventor: McMaster, et al. | Patent Number: 6821998

Compounds useful in therapy
Inventor: Gibson, et al. | Patent Number: 6812236

Analogs of cocaine
Inventor: Kozikowski, et al. | Patent Number: 6806281

Urea compounds, process for producing the same and use thereof
Inventor: Kurasawa, et al. | Patent Number: 6787650

Crystalline 3-{4-methyl-3-[methyl-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-amino]-piperidin-1 -yl}-3-oxo-propionitrile citrate
Inventor: Jacobelli | Patent Number: 6787563

N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
Inventor: Ko, et al. | Patent Number: 6780857

Intermediates useful for the preparation of antihistaminic piperidine derivatives
Inventor: Krauss, et al. | Patent Number: 6777555

Substituted tetrahydroisoquinolines as C5a receptor modulators
Inventor: Lee, et al. | Patent Number: 6777422

Melanin concentrating hormone receptor ligands
Inventor: Bakthavatchalam, et al. | Patent Number: 6753336

Arylpiperidinol and arylpiperidine derivatives and pharmaceuticals containing the same
Inventor: Annoura, et al. | Patent Number: 6706734

Inhibitors of protein isoprenyl transferases
Inventor: Sebti, et al. | Patent Number: 6693123

Sulfonamide derivatives as 5-HT7 receptor antagonists
Inventor: Lovell | Patent Number: 6660751

1-Phenacyl-3-phenyl-3-(piperidylethyl)piperidine derivatives, process for the preparation thereof and pharmaceutical compositions containing them
Inventor: Ducoux, et al. | Patent Number: 6642233

.alpha.1b-adrenergic receptor antagonists
Inventor: Hayashi, et al. | Patent Number: 6642228

Substituted phenyl-piperidine methanone compounds
Inventor: Kolczewski, et al. | Patent Number: 6642226

Piperidine amides as modulators of chemokine receptor activity
Inventor: Duncia, et al. | Patent Number: 6638950

Preferentially substituted calcium channel blockers
Inventor: Snutch | Patent Number: 6617322

N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
Inventor: Ko, et al. | Patent Number: 6605623

N-cyclopentyl modulators of chemokine receptor activity
Inventor: Finke, et al. | Patent Number: 6593346

3,3-Biarylpiperidine and 2,2-biarylmorpholine derivatives
Inventor: Liras, et al. | Patent Number: 6586431

Leukotriene B4 antagonist compounds and method for treatment
Inventor: Nakai, et al. | Patent Number: 6583177

Sulfonylcarboxamide derivatives, process for their preparation and their use as pharmaceuticals
Inventor: Kirsch, et al. | Patent Number: 6552048

Cyclopentyl modulators of chemokine receptor activity
Inventor: Yang, et al. | Patent Number: 6545023

Oxamic acids and derivatives as thyroid receptor ligands
Inventor: Chiang, et al. | Patent Number: 6545018

Inhibitors of p38-a kinase
Inventor: Goehring, et al. | Patent Number: 6541477

Cyclopentyl modulators of chemokine receptor activity
Inventor: Finke, et al. | Patent Number: 6538002

2-substituted piperidine analogs and their use as subtype-selective NMDA receptor antagonists
Inventor: Bigge, et al. | Patent Number: 6534525

Subtype-selective NMDA receptor ligands and the use thereof
Inventor: Bigge, et al. | Patent Number: 6534522

Compounds with activity on muscarinic receptors
Inventor: Brann, et al. | Patent Number: 6528529

N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
Inventor: Ko, et al. | Patent Number: 6525069

N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
Inventor: Ko, et al. | Patent Number: 6521592

Compounds
Inventor: Baxter, et al. | Patent Number: 6518286

Compounds
Inventor: Baxter, et al. | Patent Number: 6518286

N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
Inventor: Ko, et al. | Patent Number: 6492400

Partially saturated calcium channel blockers
Inventor: Snutch | Patent Number: 6492375

N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
Inventor: Ko, et al. | Patent Number: 6486180

Intermediates useful for the preparation of antihistaminic piperidine derivatives
Inventor: Krauss, et al. | Patent Number: 6479663

Method for symmetrically and asymmetrically disubstituting carboxylic acid amides with organotitanates and grignard reagents
Inventor: Buchholz, et al. | Patent Number: 6479661

Process for production of piperidine derivatives
Inventor: D'Ambra, et al. | Patent Number: 6458958

Arylpiperidinol and arylpiperidine derivatives and drugs containing the same
Inventor: Annoura, et al. | Patent Number: 6455549

Process for the preparation of hydroxamic acid derivatives
Inventor: Stabler | Patent Number: 6452010

4-substituted piperidine analogs and their use as subtype selective NMDA receptor antagonists
Inventor: Bigge, et al. | Patent Number: 6448270

4-substituted piperidine analogs and their use as subtype selective NMDA receptor antagonists
Inventor: Bigge, et al. | Patent Number: 6448270

Process for production of piperidine derivatives
Inventor: D'Ambra, et al. | Patent Number: 6444824

N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
Inventor: Ko, et al. | Patent Number: 6444686

Intermediates useful for the preparation of antihistaminic piperidine derivatives
Inventor: Krauss, et al. | Patent Number: 6441179

Biocidal benzylbiphenyl derivatives
Inventor: Meerpoel, et al. | Patent Number: 6440440

Cyclopentyl modulators of chemokine receptor activity
Inventor: Finke, et al. | Patent Number: 6432981

Aminobutyric acid derivatives
Inventor: Takahashi, et al. | Patent Number: 6420427

Anilide derivative, production and use thereof
Inventor: Shiraishi, et al. | Patent Number: 6413947

Preferentially substituted calcium channel blockers
Inventor: Snutch | Patent Number: 6387897

Chiral amino alcohols and process for preparation of same
Inventor: Goralski, et al. | Patent Number: 6362373

N-cyclopentyl modulators of chemokine receptor activity
Inventor: Finke, et al. | Patent Number: 6358979

N-cyclopentyl modulators of chemokine receptor activity
Inventor: Finke, et al. | Patent Number: 6358979

Trifluoromethyl ketone analogs as selective cPLA2 inhibitors
Inventor: Banville, et al. | Patent Number: 6350892

Intermediates useful for the preparation of antihistaminic piperidine derivatives
Inventor: Krauss, et al. | Patent Number: 6348597

Sulfonylcarboxamide derivatives, process for their preparation and their use as pharmaceuticals
Inventor: Kirsch, et al. | Patent Number: 6342512

Sulfonylcarboxamide derivatives, process for their preparation and their use as pharmaceuticals
Inventor: Kirsch, et al. | Patent Number: 6342512

Intermediates useful for the preparation of antihistaminic piperidine derivatives
Inventor: Krauss, et al. | Patent Number: 6340761

N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
Inventor: Ko, et al. | Patent Number: 6331541

Oxamic acids and derivatives as thyroid receptor ligands
Inventor: Chiang, et al. | Patent Number: 6326398

Ethanesulfonyl-piperidine derivatives
Inventor: Alanine, et al. | Patent Number: 6310213

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