Patent International Class: C07C 311/19

«1

Human adam-10 inhibitors
Inventor: Brown, et al. | Patent Number: 7951972

Human ADAM-10 inhibitors
Inventor: Brown, et al. | Patent Number: 7498358

N-cyclohexylaminocarbonyl benzensulfonmide derivatives
Inventor: Sahoo, et al. | Patent Number: 7319170

Amino acid derivatives, method for production thereof and pharmaceutical compositions comprising said derivative
Inventor: De Nanteuil, et al. | Patent Number: 7265220

Sulfonylaminocarboxylic acids
Inventor: Thorwart, et al. | Patent Number: 7160903

Derivatives of n-(arylsulfonyl)beta-aminoacids comprising a substituted aminomethyl group, the preparation method thereof and the pharmaceutical compositions containing same
Inventor: Ferrari, et al. | Patent Number: 7157454

Sulfonamide derivatives
Inventor: Hart, et al. | Patent Number: 7109203

Hydrophobic polyamine analogs and methods for their use
Inventor: Burns, et al. | Patent Number: 6963010

Preparation and purification of antiviral disulfonic acid disodium salt
Inventor: Iera, et al. | Patent Number: 6960686

Sulfonated amino acid derivatives and metalloproteinase inhibitors containing the same
Inventor: Wantanabe, et al. | Patent Number: 6919375

Method of inhibiting matrix metalloproteinases
Inventor: O'Brien, et al. | Patent Number: 6906092

MMP-12 inhibitors
Inventor: Hori, et al. | Patent Number: 6897237

Carbamic acid compounds comprising a sulfonamide linkage as HDAC inhibitors
Inventor: Watkins, et al. | Patent Number: 6888027

Compounds and methods for the treatment or prevention of Flavivirus infections
Inventor: Chan Chun Kong, et al. | Patent Number: 6887877

Sulfonated amino acid derivatives and metalloproteinase inhibitors containing the same
Inventor: Watanabe, et al. | Patent Number: 6881727

Small molecule inhibitors of caspases
Inventor: Choong, et al. | Patent Number: 6878743

Polyamine analogues as cytotoxic agents
Inventor: Burns | Patent Number: 6872852

.alpha.- and .beta.-amino acid hydroxyethylamino sulfonamides useful as retroviral protease inhibitors
Inventor: Vazquez, et al. | Patent Number: 6846954

Sulfonated amino acid derivatives and metalloproteinase inhibitors containing the same
Inventor: Wantanabe, et al. | Patent Number: 6838483

Pyrimidine compounds and derivatives thereof
Inventor: Ruminski, et al. | Patent Number: 6831199

Preparation and purification of antiviral disulfonic acid disodium salt
Inventor: Iera, et al. | Patent Number: 6806366

Analgesic compounds, their synthesis and pharmaceutical compositions containing them
Inventor: Sunkel, et al. | Patent Number: 6806291

Diaminopropionic acid derivatives
Inventor: Fotouhi, et al. | Patent Number: 6803384

FXR modulators
Inventor: Houze, et al. | Patent Number: 6777446

Process for preparing optically active amino acid derivatives
Inventor: Sugawara, et al. | Patent Number: 6720449

Caspase inhibitors and the use thereof
Inventor: Cai, et al. | Patent Number: 6716818

Cyclic derivatives as modulators of chemokine receptor activity
Inventor: Cherney | Patent Number: 6706712

Prodrugs activated by targeted catalytic proteins
Inventor: von Borstel, et al. | Patent Number: 6702705

Compounds and compositions for delivering active agents
Inventor: Leone-Bay, et al. | Patent Number: 6699467

.alpha.-hydroxyarylbutanamine inhibitors of aspartyl protease
Inventor: Or, et al. | Patent Number: 6696494

Beta disubstituted metalloprotease inhibitors
Inventor: Pikul, et al. | Patent Number: 6696456

2'-substituted 1,1'-biphenyl-2-carboxamides, process for their preparation, their use as medicaments, and pharmaceutical preparations comprising them
Inventor: Brendel, et al. | Patent Number: 6686395

Urokinase inhibitors
Inventor: Wilhelm, et al. | Patent Number: 6680320

HIV protease inhibitors based on amino acid derivatives
Inventor: Stranix, et al. | Patent Number: 6677367

Biphenyl and biphenyl-analogous compounds as integrin antagonists
Inventor: Albers, et al. | Patent Number: 6677360

Biphenyl and biphenyl-analogous compounds as integrin antagonists
Inventor: Albers, et al. | Patent Number: 6677360

HIV protease inhibitors based on amino acid derivatives
Inventor: Stranix, et al. | Patent Number: 6656965

Polyamine analogues as therapeutic and diagnostic agents
Inventor: Vermeulin, et al. | Patent Number: 6646149

Compounds and compositions for delivering active agents
Inventor: Leone-Bay, et al. | Patent Number: 6623731

Method of inhibiting matrix metalloproteinases
Inventor: O'Brien, et al. | Patent Number: 6620835

Process for preparation of optically active N-substituted azetidine-2-carboxylic acids
Inventor: Nagashima | Patent Number: 6617461

Inhibitors of aspartyl protease
Inventor: Hale, et al. | Patent Number: 6617350

Method for the synthesis of compounds of formula I and their uses thereof
Inventor: Mjalli, et al. | Patent Number: 6613801

N-(arylsulphonyl) amino acid derivatives
Inventor: Ferrari, et al. | Patent Number: 6610882

N-(arylsulphonyl) amino acid derivatives
Inventor: Ferrari, et al. | Patent Number: 6610882

HIV protease inhibitors based on amino acid derivatives
Inventor: Stranix, et al. | Patent Number: 6610689

HIV protease inhibitors based on amino acid derivatives
Inventor: Stranix, et al. | Patent Number: 6608100

.beta.-phenylalanine derivatives as integrin antagonists
Inventor: Schoop, et al. | Patent Number: 6589972

Preparation of phosphatase inhibitors
Inventor: Burgess, et al. | Patent Number: 6586467

Method for synthesis of .alpha.-sulfonamido amide, carboxylic acid and hydroxamic acid derivatives
Inventor: Campian, et al. | Patent Number: 6583318

Substituted aminoalkylamide derivatives as antagonists of follicle stimulating hormone
Inventor: Coats, et al. | Patent Number: 6583179

Peptide analogs as irreversible interleukin-1.beta. protease inhibitors
Inventor: Dolle, et al. | Patent Number: 6576614

Synthesis of .alpha.,.beta.-substituted amino amides, esters, and acids
Inventor: Sharpless, et al. | Patent Number: 6573387

Integrin antagonists
Inventor: Scarborough, et al. | Patent Number: 6552079

Angiogenesis inhibitor
Inventor: Fukiage, et al. | Patent Number: 6551999

Benzenesulphonamide compounds
Inventor: Lavielle, et al. | Patent Number: 6541471

2'-Substituted 1,1'-biphenyl-2-carboxamides, processes for their preparation, their use as medicaments, and pharmaceutical preparations comprising them
Inventor: Brendel, et al. | Patent Number: 6531495

Urea derivatives as HIV aspartyl protease inhibitors
Inventor: Stranix, et al. | Patent Number: 6528532

N-substituted arylsulfonylamino hydroxamic acids useful as inhibitors of c-proteinase and for treating or preventing disorders related to unregulated collagen production
Inventor: Ho | Patent Number: 6506936

HIV protease inhibitors based on amino acid derivatives
Inventor: Stranix, et al. | Patent Number: 6506786

Peptidyl-2-amino-1-hydroxyalkanesulfonic acid cysteine protease inhibitors
Inventor: Tao, et al. | Patent Number: 6500802

Succinoylamino hydroxyethylamino sulfonamides useful as retroviral protease inhibitors
Inventor: Vazquez, et al. | Patent Number: 6469207

Amino acid derivatives as HIV aspartyl protease inhibitors
Inventor: Bouzide, et al. | Patent Number: 6455587

Sulfonylaminocarboxylic acids
Inventor: Thorwart, et al. | Patent Number: 6451824

Sulfonylaminocarboxylic acids
Inventor: Thorwart, et al. | Patent Number: 6451824

Sulfonated amino acid derivatives and metalloproteinase inhibitors containing the same
Inventor: Wantanabe, et al. | Patent Number: 6441021

N-(arylsulphonyl) amino acid derivatives, process for their preparation and pharmaceutical compositions containing them
Inventor: Ferrari, et al. | Patent Number: 6433185

Amphiphilic polyamine compounds
Inventor: Felgner, et al. | Patent Number: 6433017

Compounds and compositions for delivering active agents
Inventor: Leone-Bay, et al. | Patent Number: 6428780

Therapeutic or prophylactic agent for glomerulopathy
Inventor: Kurihara, et al. | Patent Number: 6423729

Biphenyl and biphenyl-analogous compounds as integrin antagonists
Inventor: Albers, et al. | Patent Number: 6420396

Sulfonylamino derivatives which inhibit matrix-degrading metalloproteinases
Inventor: Kukkola, et al. | Patent Number: 6410580

Method of treating disease with sulfonylamino acid derivatives
Inventor: Sakaki, et al. | Patent Number: 6403644

Amine and amide derivatives as ligands for the neuropeptide Y Y5 receptor useful in the treatment of obesity and other disorders
Inventor: Dax, et al. | Patent Number: 6380224

Substituted diaminocarboxylic acids
Inventor: Thorwart, et al. | Patent Number: 6355673

Substituted diaminocarboxylic acids
Inventor: Thorwart, et al. | Patent Number: 6355673

Caspase inhibitors and the use thereof
Inventor: Cai, et al. | Patent Number: 6355618

Aminohydroxylation of Olefins
Inventor: Sharpless, et al. | Patent Number: 6350905

Aminobutyric acid fungicides
Inventor: Cohen, et al. | Patent Number: 6348614

Oxime ethers as IIb/IIa antagonists
Inventor: Olson, et al. | Patent Number: 6348504

Amphiphilic polyamide compounds
Inventor: Felgner, et al. | Patent Number: 6348499

Peptidyl-2-amino-1-hydroxyalkanesulfonic acid cysteine protease inhibitors
Inventor: Tao, et al. | Patent Number: 6348448

Compounds and compositions for delivering active agents
Inventor: Leone-Bay, et al. | Patent Number: 6346242

Tyrosine alkoxyguanidines as integrin inhibitors
Inventor: Tomczuk, et al. | Patent Number: 6344484

N-arylsulfonylamino acid omega-amides
Inventor: Schwab, et al. | Patent Number: 6335333

Diaminopropionic acid derivatives
Inventor: Fotouhi, et al. | Patent Number: 6331640

Inhibitors of aspartyl protease
Inventor: Hale, et al. | Patent Number: 6319946

Sulfonamide interleukin-1.beta. converting enzyme inhibitors
Inventor: Albrecht, et al. | Patent Number: 6316415

N-(arylsulfonyl) amino acid derivatives, process for their preparation and pharmaceutical compositions containing them
Inventor: Ferrari, et al. | Patent Number: 6313120

Process to prepare taxol
Inventor: Wuts, et al. | Patent Number: 6307064

.beta.-phenylalanine derivatives as integrin antagonists
Inventor: Schoop, et al. | Patent Number: 6291503

Sulfonylamino acid and sulfonylamino hydroxamic acid derivatives
Inventor: Kukkola, et al. | Patent Number: 6277987

Cyclic amino acid derivatives as cell adhesion inhibitors
Inventor: Chang, et al. | Patent Number: 6271252

Hydrazide compounds
Inventor: Monge Vega, et al. | Patent Number: 6271247

Prodrugs activated by targeted catalytic proteins
Inventor: von Borstel, et al. | Patent Number: 6258360

Para-substituted phenylene derivatives
Inventor: Chen, et al. | Patent Number: 6251944

Integrin antagonists
Inventor: Scarborough, et al. | Patent Number: 6245809

Substituted .beta.-amino acid inhibitors of methionine aminopeptidase-2
Inventor: Craig, et al. | Patent Number: 6242494

Compounds
Inventor: Faller | Patent Number: 6242467

Benzenesulfonamide compounds
Inventor: Ohuchida, et al. | Patent Number: 6235777

«1