Patent International Class: A61P 25/18

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Substituted thieno[2,3-d]pyrimidines as AMPA modulators
Inventor: Gallagher, et al. | Patent Number: 8129397

Therapeutic agents 713
Inventor: Johansson, et al. | Patent Number: 8110566

Triazole compounds suitable for treating disorders that respond to modulation of the dopamine D.sub.3 receptor
Inventor: Unger, et al. | Patent Number: 8101754

Quetiapine salts and their polymorphs
Inventor: Dixit, et al. | Patent Number: 8101597

Substituted pyrazolo [1,5-a] pyrimidines as metabotropic glutamate antagonists
Inventor: Gatti McArthur, et al. | Patent Number: 8093263

Polysubstituted derivatives of 6-heteroarylimidazo[1,2-a]pyridines, and preparation and therapeutic use thereof
Inventor: De Peretti, et al. | Patent Number: 8088765

Dialkylamino alkyl esters of pivagabine as medicaments for the treatment of central nervous system disorders
Inventor: Rafferty | Patent Number: 8080548

Carbocyclic GlyT-1 receptor antagonists
Inventor: Kolczewski, et al. | Patent Number: 8080541

2-cyanophenyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine compounds, compositions and uses thereof
Inventor: Wei, et al. | Patent Number: 8076345

Substituted pyridazine derivatives
Inventor: Hudkins, et al. | Patent Number: 8076331

Acetylenyl-pyrazolo-pyrimidine derivatives
Inventor: Gatti McArthur, et al. | Patent Number: 8063048

Pyridazine compounds and methods
Inventor: Watterson, et al. | Patent Number: 8063047

Methods of treating disease with nitric oxide (NO)-releasing polymers and soluble no-releasing nitrosamines
Inventor: Oh-Lee, et al. | Patent Number: 8062656

6-cyclylmethyl- and 6-alkylmethyl pyrazolo[3,4-D]pyrimidines, methods for their preparation and methods for their use to treat impairments of perception, concentration learning and/or memory
Inventor: Hendrix, et al. | Patent Number: 8044060

Crystallization process of quetiapine hemifumarate
Inventor: Rummakko, et al. | Patent Number: 8044038

Modified release compositions of milnacipran
Inventor: Hirsh, et al. | Patent Number: 8021687

Salt forms of (2S)-(4E)-N-methyl-5-[3-(5-isopropoxypyridin)y1]-4-penten 2-amine
Inventor: Ericsson, et al. | Patent Number: 8017785

Pyrimidin-2-one compounds and their use as dopamine D.sub.3 receptor ligands
Inventor: Geneste, et al. | Patent Number: 8008488

Arylpiperazine derivatives and uses thereof
Inventor: Carter, et al. | Patent Number: 7998963

Compounds having affinity for dopamine D3 receptor and uses thereof
Inventor: Bonanomi, et al. | Patent Number: 7989444

Process for the preparation of olanzapine
Inventor: Kovanyine Lax, et al. | Patent Number: 7981884

5HT.sub.2C receptor modulators
Inventor: Smith, et al. | Patent Number: 7977329

Pharmaceutical composition of quetiapine fumarate
Inventor: Jansen | Patent Number: 7959948

Polymorphs of olanzapine hydrochloride
Inventor: Petho, et al. | Patent Number: 7951798

3-(1,2,4-triazol-3-ylalkyl) azabicyclo (3.1.0) hexane derivatives as modulators of dopamine D3 receptors
Inventor: Bonanomi, et al. | Patent Number: 7947683

Aminoazacyclyl-3-sulfonylindazoles as 5-hydroxytryptamine-6 ligands
Inventor: Haydar, et al. | Patent Number: 7939520

Pyrrolo[2,3-d]pyrimidine derivatives substituted with a cyclic amino group
Inventor: Nakazato, et al. | Patent Number: 7932259

Olanzapine pamoate dihydrate
Inventor: Bush | Patent Number: 7932249

Substituted 2,5-dihydro-3H-pyrazolo[4,3-C]pyridazin-3-one derivatives, preparation thereof and therapeutic use of the same
Inventor: Congy, et al. | Patent Number: 7915258

Levodopa prodrug mesylate, compositions thereof, and uses thereof
Inventor: Xiang, et al. | Patent Number: 7893105

Compositions useful as inhibitors of GSK-3
Inventor: Forster, et al. | Patent Number: 7872129

Carbonylbenzoxazine compounds for enhancing glutamatergic synaptic responses
Inventor: Rogers, et al. | Patent Number: 7799913

Compounds capable of activating cholinergic receptors
Inventor: Caldwell, et al. | Patent Number: 7790757

Thienopyrimidine compounds and uses thereof
Inventor: Giordanetto, et al. | Patent Number: 7723331

Acetylenyl-pyrazolo-pyrimidine derivatives
Inventor: Gatti McArthur, et al. | Patent Number: 7718661

Dealkylated derivatives of pyrrolo[2,1-b]benzothiazepines with atypical antipsychotic activity
Inventor: Carminati, et al. | Patent Number: 7713956

Haloperidol analogs
Inventor: Ablordeppey, et al. | Patent Number: 7700587

Pyrazole compounds useful as protein kinase inhibitors
Inventor: Bebbington, et al. | Patent Number: 7691853

Substituted 1(2H)-phthalazinones and pharmaceutical compositions thereof
Inventor: Upasani, et al. | Patent Number: 7652006

Cyclic amine compound
Inventor: Kumagai, et al. | Patent Number: 7601734

Triazol[4,5-d] pyramidine derivatives and their use as purinergic receptor antagonists
Inventor: Gillespie, et al. | Patent Number: 7589097

Therapeutic agents
Inventor: Cheng | Patent Number: 7576095

Certain thienopyrimidine derivatives as phosphodiesterase 10 inhibitors
Inventor: Liu, et al. | Patent Number: 7576080

Substituted sulfonamide compounds useful for the prophylaxis and treatment of conditions relating to obesity, type II diabetes and/or disorders of the central nervous system
Inventor: Bremberg, et al. | Patent Number: 7566715

Substituted pyrrolo[3,2-d]pyrimidine derivatives
Inventor: Tsutsumi, et al. | Patent Number: 7557113

Substituted 8'-pyri(MI)dinyl-dihydrospiro-[cycloalkylamine]-pyrimido[1,2-a]pyrimidin-- 6-one derivatives
Inventor: Chereze, et al. | Patent Number: 7547705

Conjugated psychotropic drugs and uses thereof
Inventor: Nudelman, et al. | Patent Number: 7544681

Triazine derivatives, their preparation and therapeutic application thereof
Inventor: Benedetti, et al. | Patent Number: 7517881

5HT.sub.2c receptor modulators
Inventor: Smith, et al. | Patent Number: 7514422

Compounds as metabotropic glutamate receptor antagonists
Inventor: McArthur, et al. | Patent Number: 7504404

Benzoxazepine derivatives and their use as AMPA receptor stimulators
Inventor: Grove, et al. | Patent Number: 7504390

Indolylalkylamine metabolites as 5-hydroxytryptamine-6 ligands
Inventor: Wang, et al. | Patent Number: 7498327

Compositions useful as inhibitors of GSK-3
Inventor: Forster, et al. | Patent Number: 7491730

Amino substituted diaryl[a,d]cycloheptene analogs as muscarinic agonists and methods of treatment of neuropsychiatric disorders
Inventor: Ek, et al. | Patent Number: 7491715

Substituted phenyl methanones
Inventor: Jolidon, et al. | Patent Number: 7442710

Tetrahydrobenzazepine derivatives useful as modulators of dopamine D3 receptors (antipsychotic agents)
Inventor: Hadley, et al. | Patent Number: 7429579

Substituted pyrimidines
Inventor: Kopka, et al. | Patent Number: 7405221

Triazolo [4,5-d] pyrimidine derivatives and their use as purinergic receptor antagonists
Inventor: Gillespie, et al. | Patent Number: 7405219

Phosphodiesterase 4 inhibitors
Inventor: Tehim, et al. | Patent Number: 7332486

Crystal forms, methods for their preparation and method for preparation of olanzapine
Inventor: Dolitzky, et al. | Patent Number: 7323459

COMT inhibitors for the treatment of depression and impaired cognition
Inventor: Diederich, et al. | Patent Number: 7319101

Compounds Capable of Activating Cholinergic Receptors
Inventor: Caldwell, et al. | Patent Number: 7307092

Process of preparation of olanzapine form I
Inventor: Patel, et al. | Patent Number: 7297789

Cannabinoid receptor ligands and uses thereof
Inventor: Griffith, et al. | Patent Number: 7268133

Compositions for the treatment of neurological disorders
Inventor: Mann | Patent Number: 7261907

Preparation of risperidone
Inventor: Krochmal, et al. | Patent Number: 7256195

Treatment of aging disorders in humans
Inventor: Rodriguez | Patent Number: 7256184

Pyrimidine compounds and their use
Inventor: Nilsson | Patent Number: 7247633

Substituted indoles and their use as integrin antagonists
Inventor: Lu, et al. | Patent Number: 7241789

Lactam derivatives as antagonists for human 11cby receptors
Inventor: Armstrong, et al. | Patent Number: 7220777

Substituted imidazotriazines
Inventor: Hendrix, et al. | Patent Number: 7202243

[1,4]Diazepino[6,7,1-ij]quinoline derivatives as antipsychotic and antiobesity agents
Inventor: Ramamoorthy | Patent Number: 7129237

Adenosine A2a receptor antagonists
Inventor: Matasi, et al. | Patent Number: 7041666

Positive allosteric AMPA receptor modulators (PAARM), processes for preparing them, and their use as pharmaceutical compositions
Inventor: Ceci, et al. | Patent Number: 7026475

Indolylalkylamine derivatives as 5-hydroxytryptamine-6 ligands
Inventor: Cole, et al. | Patent Number: 7022701

Pharmaceutical compositions containing new polymorphic forms of olanzapine and uses thereof
Inventor: Hamied, et al. | Patent Number: 7022698

[1,4]Diazocino[7,8,1-hi]indole derivatives as antipsychotic and antiobesity agents
Inventor: Gao, et al. | Patent Number: 7012089

Pharmaceutical compositions containing lithium carbonate
Inventor: Tarro | Patent Number: 6989159

Fluorobenzamides and uses thereof
Inventor: Jolidon, et al. | Patent Number: 6951884

Dihydro-benzo[b][1,4]diazepin-2-one derivatives
Inventor: Adam, et al. | Patent Number: 6949542

Method of treating psychosis in a patient
Inventor: Chern, et al. | Patent Number: 6946470

Benzoxazinone derivatives, their preparation and use
Inventor: Johnson, et al. | Patent Number: 6939871

Azaindoles having serotonin receptor affinity
Inventor: Edwards, et al. | Patent Number: 6916818

Adenosine A2a receptor antagonists
Inventor: Boyle, et al. | Patent Number: 6916811

Pharmaceutical compositions comprising cyclic glycerophosphates and analogs thereof for promoting neural cell differentiation
Inventor: Shinitzky | Patent Number: 6914056

Antipsychotic cyclic N-aralkylamines
Inventor: Boigegrain, et al. | Patent Number: 6908914

Crystalline form I of 2-methyl-4-(4-menthyl-1-piperazinyl) 10H thieno [2,3-b][1,5]benzodiazepine
Inventor: Chhabada, et al. | Patent Number: 6906062

Serotonergic agents with long-acting in vivo effects
Inventor: Childers, et al. | Patent Number: 6894053

Atypical antipsychotic agents having low affinity for the D2 receptor
Inventor: Kapur, et al. | Patent Number: 6890919

Tetracyclic azepinoindole compounds
Inventor: Hester, et al. | Patent Number: 6875762

Method of treating bipolar disorders using deuterium-substituted carbonate
Inventor: Bell | Patent Number: 6872408

N-substituted 1,2,4,5-tetrahydro-1H-benzo[d]azepine compounds
Inventor: Fu | Patent Number: 6861420

Substituted indoles and their use as integrin antagonists
Inventor: Lu, et al. | Patent Number: 6855722

Protein kinase inhibitors and uses thereof
Inventor: Moon, et al. | Patent Number: 6825190

Antipsychotic aminomethyl derivatives of 7,8-dihydro-3H-6,9-dioxa-2,3-diaza-cyclopenta[a]naphthalene
Inventor: Tran, et al. | Patent Number: 6800641

4-piperazinylindole derivatives with 5-HT6 receptor affinity
Inventor: Briggs, et al. | Patent Number: 6790848

Substituted pyrroloquinolines and pyridoquinolines as serotinin agonists and antagonists
Inventor: Fevig, et al. | Patent Number: 6777406

Indolylalkylamine derivatives as 5-hydroxytryptamine-6 ligands
Inventor: Cole, et al. | Patent Number: 6770642

Pyrimidin-4-one compounds
Inventor: Lavielle, et al. | Patent Number: 6747032

Pyrrolo[2,1-B][3,1] benzothiazepines and their use for the preparation of medicaments with antipsychotic activity
Inventor: Minetti, et al. | Patent Number: 6710041

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