Patent Class: Organic Compounds -- Part Of The Class 532-570 Series (546/199)

Description

In this series of classes, Class 546 is to be considered as anintegral part of Class 260 (after subclass 544) and follows theschedule hierarchy retaining all pertinent definitions and classlines of Class 260.

«1...

Piperidine derivative or salt thereof
Inventor: Hachiya, et al. | Patent Number: 8153658

Heterocyclic compounds as factor IXA inhibitors
Inventor: Clasby, et al. | Patent Number: 8148363

Heterocyclic compounds
Inventor: Chen, et al. | Patent Number: 8143282

Aminocarbonyl-substituted 8-N-benzimidazoles, methods for their preparation and their use in pharmaceutical compositions
Inventor: DeFossa, et al. | Patent Number: 8138207

Benzimidazolone derivatives as CB2 receptor ligands
Inventor: Ando, et al. | Patent Number: 8138177

Renin inhibitors
Inventor: Jones, et al. | Patent Number: 8138168

Piperidine derivatives and their use as muscarinic receptor modulators
Inventor: Cheng, et al. | Patent Number: 8119661

2H- or 3H-benzo[e]indazol-1-yl carbamate derivatives, the preparation and therapeutic use thereof
Inventor: DuBois, et al. | Patent Number: 8114899

Indazole derivatives as kinase inhibitors for the treatment of cancer
Inventor: Bandiera, et al. | Patent Number: 8114865

Pyrazino[2,3-b]pyrazine mTOR kinase inhibitors for oncology indications and diseases associated with the mTOR/PI3K/Akt pathway
Inventor: Perrin-Ninkovic, et al. | Patent Number: 8110578

Synthetic multimerizing agents
Inventor: Holt, et al. | Patent Number: 8106191

Cytoskeletal active rho kinase inhibitor compounds, composition and use
Inventor: Lampe, et al. | Patent Number: 8071779

Amide substituted indazoles as poly(ADP-ribose)polymerase(PARP) inhibitors
Inventor: Jones, et al. | Patent Number: 8071623

Indoles
Inventor: Bissantz, et al. | Patent Number: 8071622

Benzimidazole poly(ADP ribose)polymerase inhibitors
Inventor: Gandhi, et al. | Patent Number: 8067613

Benzimidazolone and quinazolinone derivatives as agonists on human ORL1 receptors
Inventor: Den Hartog, et al. | Patent Number: 8067603

Pharmaceutical use of substituted amides
Inventor: Kilburn, et al. | Patent Number: 8053431

Thiazolyl-benzimidazoles
Inventor: Cai, et al. | Patent Number: 8044213

Use of 2h-benzimidazol-2-one, 1,3-dihydro-1-(2{4-[3-(trifluoromethyl)phenyl]-1-piperazinyl}ethyl)-and its physiologically acceptable acid addition salts
Inventor: Beck | Patent Number: 8030314

Substituted heterocyclic ethers and their use in CNS disorders
Inventor: Degnan, et al. | Patent Number: 8026257

P38 inhibitors and methods of use thereof
Inventor: Munson, et al. | Patent Number: 8026233

Indazole acrylic acid amide compound
Inventor: Yamaguchi, et al. | Patent Number: 8022059

Isoindole-imide compounds, compositions, and uses thereof
Inventor: Robarge, et al. | Patent Number: 8012997

Pharmaceutically active sulfonamide derivatives
Inventor: Arkinstall, et al. | Patent Number: 8012995

Pyrrolopyrazinyl urea kinase inhibitors
Inventor: Bamberg, et al. | Patent Number: 8012974

Indazole compounds
Inventor: Ericsson, et al. | Patent Number: 8008481

4-benzyledene-piperidin derivatives
Inventor: Borza, et al. | Patent Number: 8008326

Integrin antagonists useful as anticancer agents
Inventor: Bloxham, et al. | Patent Number: 8003806

Remedy for sleep disturbance
Inventor: Teshima, et al. | Patent Number: 8003669

Amino-substituted 8-N-benzimidazoles and methods for their use in blood sugar disorders
Inventor: Defossa, et al. | Patent Number: 8003668

CGRP receptor antagonists
Inventor: Paone, et al. | Patent Number: 7994325

Bicyclic nitrogen-containing heterocyclic compounds
Inventor: Atobe, et al. | Patent Number: 7994202

Indazole compound and pharmaceutical use thereof
Inventor: Takemiya, et al. | Patent Number: 7994196

2,4-diaminoquinazolines for spinal muscular atrophy
Inventor: Singh, et al. | Patent Number: 7985755

Compounds
Inventor: Cheng, et al. | Patent Number: 7956069

Heterocyclyl-substituted thiazoles as crop protection agents
Inventor: Cristau, et al. | Patent Number: 7943774

Aminoazacyclyl-3-sulfonylindazoles as 5-hydroxytryptamine-6 ligands
Inventor: Haydar, et al. | Patent Number: 7939520

N-substituted-azacyclylamines as histamine-3 antagonists
Inventor: Solvibile, et al. | Patent Number: 7935719

2-quinazolinone compounds and methods of use
Inventor: Hong, et al. | Patent Number: 7935709

Thienopyrazole derivative having PDE7 inhibitory activity
Inventor: Inoue, et al. | Patent Number: 7932250

Nanomolar .beta.-lactamase inhibitors
Inventor: Shoichet, et al. | Patent Number: 7928129

Substituted 6a,7,8,9-tetrahydropyrido[3,2-e]pyrrolo[1,2-a]pyrazin-6(5H)-ones
Inventor: Gangloff, et al. | Patent Number: 7928105

Substituted benzimidazole compounds with dual NOS inhibitory activity and mu opioid agonist activity
Inventor: Renton, et al. | Patent Number: 7919510

Hepatitis C virus inhibitors
Inventor: Belema, et al. | Patent Number: 7906655

Indazole derivatives
Inventor: Ishibashi, et al. | Patent Number: 7906532

Pyrazoles for the treatment of obesity and other CNS disorders
Inventor: Bennani, et al. | Patent Number: 7897634

Thiazolyl-dihydro-indazole
Inventor: McConnell, et al. | Patent Number: 7893049

Organic compounds
Inventor: Kwak, et al. | Patent Number: 7879850

Kinase inhibitors
Inventor: Bonjouklian, et al. | Patent Number: 7863310

Hydronopol substituted benzimidazolone and quinazolinone derivatives as agonists on human ORL1 receptors
Inventor: Den Hartog, et al. | Patent Number: 7851630

Substituted 4-anilinoquinazolines and their use in tumor treatment
Inventor: Huang, et al. | Patent Number: 7825245

Hexahydro-cyclooctyl pyrazole cannabinoid modulators
Inventor: Xia, et al. | Patent Number: 7825151

Modulators of muscarinic receptors
Inventor: Makings, et al. | Patent Number: 7820817

Cyclohexylimidiazole lactam derivatives as inhibitors of 11-.beta.-hydroxysteroid dehydrogenase 1
Inventor: Saeed, et al. | Patent Number: 7820659

Imidazolothiazole compounds for the treatment of disease
Inventor: Bhagwat, et al. | Patent Number: 7820657

Cyclic amides
Inventor: Schadt, et al. | Patent Number: 7816376

Compounds that are ERK inhibitors
Inventor: Deng, et al. | Patent Number: 7807672

MCH receptor antagonists
Inventor: Berthel, et al. | Patent Number: 7803816

Indol-3-yl-corbonyl-piperidin-benzoimidazol derivatives
Inventor: Bissantz, et al. | Patent Number: 7803815

Indoles
Inventor: Bissantz, et al. | Patent Number: 7799923

Derivatives of N-[phenyl(alkylpiperidine-2-yl)methyl]benzamide, preparation method thereof and application of same in therapeutics
Inventor: Dargazanli, et al. | Patent Number: 7790753

Azinyl-3-sulfonylindazole derivatives as 5-hydroxytryptamine-6 ligands
Inventor: Elokdah, et al. | Patent Number: 7790751

Monocyclic and bicyclic compounds and methods of use
Inventor: Zhang, et al. | Patent Number: 7790726

Pyrroloquinoxalinone inhibitors of poly(ADP-ribose)polymerase
Inventor: Giranda, et al. | Patent Number: 7790721

Tetrahydro-cyclopentyl pyrazole cannabinoid modulators
Inventor: Liotta, et al. | Patent Number: 7790718

Organic compounds
Inventor: Herold, et al. | Patent Number: 7790715

Substituted 2-phenylbenzimidazoles, the production thereof and their use
Inventor: Lubisch, et al. | Patent Number: 7781596

Benzimidazolone compounds having 5-HT4 receptor agonistic activity
Inventor: Katsu, et al. | Patent Number: 7776885

Diaminoalkane aspartic protease inhibitors
Inventor: Baldwin, et al. | Patent Number: 7754737

Benzimidazole-derivatives as factor Xa inhibitors
Inventor: Nazare, et al. | Patent Number: 7741341

Benzimidazolone carboxylic acid derivatives
Inventor: Ando, et al. | Patent Number: 7737163

Alkyl-and piperidine-substituted benzimidazole derivatives
Inventor: Anderskewitz, et al. | Patent Number: 7723360

Substituted-3-sulfonylindazole derivatives as 5-hydroxytryptamine-6 ligands
Inventor: Elokdah, et al. | Patent Number: 7723329

Imidazo[1,2-A]pyridine anxiolytics
Inventor: Fang, et al. | Patent Number: 7723324

NK1 antagonists
Inventor: Shah, et al. | Patent Number: 7709641

Pyrrolo-quinoxalinone derivatives as antibacterials
Inventor: Jones, et al. | Patent Number: 7709483

Benzimidazolone carboxylic acid derivatives
Inventor: Ando, et al. | Patent Number: 7705020

Bicyclic heteroaromatic compounds
Inventor: Leach | Patent Number: 7705005

Fused heteroaryl derivatives for use as p38 kinase inhibitors in the treatment of I.A. rheumatoid arthritis
Inventor: Campos, et al. | Patent Number: 7687532

N-linked aryl heteroaryl inhibitors of LTA4H for treating inflammation
Inventor: Sandanayaka, et al. | Patent Number: 7674802

Heteroindanes: a new class of potent cannabimimetic ligands
Inventor: Makriyannis, et al. | Patent Number: 7666867

Indazole having analgesic activity
Inventor: Alisi, et al. | Patent Number: 7662836

Unsaturated mTOR inhibitors
Inventor: Crew, et al. | Patent Number: 7659274

Compositions useful as inhibitors of protein kinases
Inventor: Binch, et al. | Patent Number: 7652135

2-(R)-(4-fluoro-2-methyl-phenyl)-4-(S)-((8aS)-6-oxo-hexahydro-pyrrolo[1,2-- a]-pyrazin-2-yl)-piperidine-1-carboxylic acid [1-(R)-3,5-bis-trifluoromethyl-phenyl)-ethyl]-methylamide maleate and pharmaceutical compositions thereof
Inventor: Alvaro, et al. | Patent Number: 7652012

Indazolamides with analgesic activity
Inventor: Alisi, et al. | Patent Number: 7632849

Intermediate for the preparation of paliperidone
Inventor: Hu, et al. | Patent Number: 7629469

Octahydro-pyrrolo[3,4-c]pyrrole CCR5 receptor antagonists
Inventor: Lemoine, et al. | Patent Number: 7625905

Substituted bis aryl and heteroaryl compounds as selective 5HT.sub.2A antagonists
Inventor: Eastwood, et al. | Patent Number: 7625889

Benzimidazole thiophene compounds
Inventor: Kuntz, et al. | Patent Number: 7615643

Polymorph of 4-[2-[4-[1-(2-ethoxyethyl)-1H-benzimidazole-2-yl]-1-piperidinyl]ethyl]-.a- lpha..alpha.-dimethyl-benzeneacetic acid
Inventor: Orjales Venero, et al. | Patent Number: 7612095

IGF-1R inhibitor
Inventor: Kanda, et al. | Patent Number: 7605272

Compounds having activity as inhibitors of apoptosis
Inventor: Cottam, et al. | Patent Number: 7601846

Cyclic amine compound
Inventor: Kumagai, et al. | Patent Number: 7601734

Benzimidazole thiophene compounds
Inventor: Cheung, et al. | Patent Number: 7595330

Benzimidazolone carboxylic acid derivatives
Inventor: Ando, et al. | Patent Number: 7595329

Indane compounds as CCR5 antagonists
Inventor: Youngman, et al. | Patent Number: 7589204

1-Heterocyclylalkyl-3-sulfonylindole or -indazole derivatives as 5-hydroxytryptamine-6 ligands
Inventor: Bernotas, et al. | Patent Number: 7589108

Pyrrolo[3,4-c]pyrazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them
Inventor: Fancelli, et al. | Patent Number: 7582628

Propane-1, 3-dione derivative
Inventor: Hirano, et al. | Patent Number: 7569688

«1...