Patent Class: Organic Compounds -- Part Of The Class 532-570 Series (546/139)

Description

In this series of classes, Class 546 is to be considered as anintegral part of Class 260 (after subclass 544) and follows theschedule hierarchy retaining all pertinent definitions and classlines of Class 260.

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5-HT7 receptor antagonists
Inventor: Torrens Jover, et al. | Patent Number: 8148397

Process of producing bleach boosters
Inventor: Voelkel, et al. | Patent Number: 8129531

Bicyclic compounds with kinase inhibitory activity
Inventor: Calderwood, et al. | Patent Number: 8110687

Process for the preparation of onium salts with a tetrafluoroborate anion having a reduced halide content
Inventor: Ignatyev, et al. | Patent Number: 8101749

Histone deacetylase inhibitors and methods of use thereof
Inventor: Kozikowski, et al. | Patent Number: 8067600

Kappa opioid receptor ligands
Inventor: Carroll, et al. | Patent Number: 8048895

2-(aryloxy) acetamide factor VIIa inhibitors useful as anticoagulants
Inventor: Nirschl, et al. | Patent Number: 8044242

Isoxazoline derivative and novel process for its preparation
Inventor: Shin, et al. | Patent Number: 8044080

Isoquinolines as IGF-1R inhibitors
Inventor: Gunzinger, et al. | Patent Number: 8044067

Benzofluoranthene compound and organic light-emitting device using the compound
Inventor: Ohrui, et al. | Patent Number: 8034944

Fused compounds that inhibit vanilloid subtype 1 (VR1) receptor
Inventor: Gomtsyan, et al. | Patent Number: 8026256

Substituted piperidines as somatostatin receptor subtype 5 (SSTR5) antagonists
Inventor: Binggeli, et al. | Patent Number: 8026255

Inhibitors of AKT (protein kinase B)
Inventor: Joseph, et al. | Patent Number: 7998977

Benzothiazepine and benzothiepine compounds
Inventor: Sasahara, et al. | Patent Number: 7973030

Sulfonamide compound
Inventor: Matsubara, et al. | Patent Number: 7964613

VR1 vanilloid receptor antagonists with a iononic substructure
Inventor: Baraldi, et al. | Patent Number: 7919624

Heterocyclic tetracyclic tetrahydrofuran derivatives as 5HT.sub.2 inhibitors in the treatment of CNS disorders
Inventor: Cid-N nez, et al. | Patent Number: 7915249

Heterocyclic modulators of PKB
Inventor: Zeng, et al. | Patent Number: 7897619

Chiral 1,8-diarylnaphthalenes, methods of making them, and their use as sensors
Inventor: Wolf, et al. | Patent Number: 7888509

Diaminothiazoles useful as Axl inhibitors
Inventor: Goff, et al. | Patent Number: 7879856

Process for production of 4-fluoroisoquinoline-5-sulfonyl halide or salt thereof
Inventor: Sakai, et al. | Patent Number: 7872136

Biphenyl compounds useful as muscarinic receptor antagonists
Inventor: Mammen, et al. | Patent Number: 7858792

Indazolyl-substituted pyrroline compounds as kinase inhibitors
Inventor: Zhang, et al. | Patent Number: 7855203

Tetrahydroisoquinoline sulfonamide derivatives, the preparation thereof, and the use of the same in therapeutics
Inventor: Diaz Martin, et al. | Patent Number: 7833999

Chromanylurea compounds that inhibit vanilloid receptor subtype 1 (VR1) receptor and uses thereof
Inventor: Gomtsyan, et al. | Patent Number: 7812019

Electron transport compound and organic light emitting device comprising the same
Inventor: Kim, et al. | Patent Number: 7811681

Derivatives of N-[phenyl(alkylpiperidine-2-yl)methyl]benzamide, preparation method thereof and application of same in therapeutics
Inventor: Dargazanli, et al. | Patent Number: 7790753

Pharmacological uses of azetidine derivatives
Inventor: Achard, et al. | Patent Number: 7741316

Dipeptidyl peptidase inhibitors
Inventor: Gwaltney, et al. | Patent Number: 7732446

Chemokine receptor antagonist and medical use thereof
Inventor: Habashita, et al. | Patent Number: 7732442

Substituted tetrahydroisoquinoline compounds, methods of making, and their use
Inventor: Miller, et al. | Patent Number: 7718672

Hepatitis C inhibitor peptide analogs
Inventor: Bailey, et al. | Patent Number: 7696242

1-isopropyl-2-oxo-1,2-dihydropyridine-3-carboxamide derivatives having 5-HT.sub.4 receptor agonistic activity
Inventor: Kato, et al. | Patent Number: 7691881

Azadecalin Glucocorticoid receptor modulators
Inventor: Clark, et al. | Patent Number: 7678813

Aminotetralin-derived urea modulators of vanilloid VR1 receptor
Inventor: Codd, et al. | Patent Number: 7678812

Aryloxyalkylcarbamate-type derivatives, preparation method thereof and use of same in therapeutics
Inventor: Abouabdellah, et al. | Patent Number: 7674805

Acetyl 2-hydroxy-1, 3-diaminoalkanes
Inventor: John, et al. | Patent Number: 7645780

Sulfonamide compound
Inventor: Yamada, et al. | Patent Number: 7618984

Inhibitors of histone deacetylase
Inventor: Delorme, et al. | Patent Number: 7595343

Vanilloid receptor ligands and their use in treatments
Inventor: Bo, et al. | Patent Number: 7579347

Benzothiazole cyclobutyl amine derivatives
Inventor: Cowart, et al. | Patent Number: 7576110

Heterocyclic compounds as inhibitors of factor VIIa
Inventor: Glunz, et al. | Patent Number: 7576098

2,5-disubstituted 3-mercaptopentanoic acid
Inventor: Polla | Patent Number: 7572817

Aryl- and heteroaryl-substituted tetrahydroisoquinolines and use thereof to block reuptake of norepinephrine, dopamine, and serotonin
Inventor: Molino, et al. | Patent Number: 7541357

Taxanes having a C10 ester substituent
Inventor: Holton | Patent Number: 7524869

Histone deacetylase inhibitors and methods of use thereof
Inventor: Kozikowski, et al. | Patent Number: 7507828

Quinoline derivatives and their use as tyrosine kinase inhibitors
Inventor: Hennequin | Patent Number: 7501516

Multicyclic sulfonamide compounds as inhibitors of histone deacetylase for the treatment of disease
Inventor: Malecha, et al. | Patent Number: 7470722

Immunosuppressant compounds and compositions
Inventor: Pan, et al. | Patent Number: 7462629

Synthesis of enantiomerically pure amino-substituted fused bicyclic rings
Inventor: McEachern, et al. | Patent Number: 7452994

7-phenyl-isoquinoline-5-sulfonylamino derivatives as inhibitors of akt (protein kinase B)
Inventor: Barda, et al. | Patent Number: 7449477

Peptidomimetic ligands for cellular receptors and ion channels
Inventor: Persons, et al. | Patent Number: 7446115

Bicyclic benzamide compound as histamine H3 receptor ligand useful in the treatment of neurological diseases
Inventor: Best, et al. | Patent Number: 7446103

Rearranged pentanols, a process for their production and their use as anti-inflammatory agents
Inventor: Rehwinkel, et al. | Patent Number: 7442794

Aryloxyalkylcarbamate-type derivatives, preparation method thereof and use of same in therapeutics
Inventor: Abouabdellah, et al. | Patent Number: 7439257

Cyanoanthranilamide derivatives and the use thereof as medicaments
Inventor: Ernst, et al. | Patent Number: 7429592

Non-imidazole aryloxyalkylamines
Inventor: Apodaca, et al. | Patent Number: 7429586

Inhibitors of Akt (protein kinase B)
Inventor: Al-Awar, et al. | Patent Number: 7414063

P2X.sub.7 receptor antagonists and their use
Inventor: Evans, et al. | Patent Number: 7408065

Protein kinase inhibitors comprising ATP mimetics conjugated to peptides or peptidomimetics
Inventor: Livnah, et al. | Patent Number: 7407939

Compounds as pharmaceutical agents
Inventor: Beight, et al. | Patent Number: 7405299

Sulfated bis-cyclic agents
Inventor: Desai, et al. | Patent Number: 7402594

Thiadiazole compounds and methods of use
Inventor: Zeng, et al. | Patent Number: 7354944

Heterocyclic retinoid compounds
Inventor: Klaus, et al. | Patent Number: 7354931

Substituted 2,3-dihydro-1h-isoindol-1-one derivatives and methods of use
Inventor: Tegley, et al. | Patent Number: 7320992

Hepatitis C virus inhibitors
Inventor: Tu, et al. | Patent Number: 7309708

5-HT.sub.7 receptor antagonists
Inventor: Curtis, et al. | Patent Number: 7276607

Substituted 2-pyrrolidine-2-yl-1H-indole compounds
Inventor: Sundermann, et al. | Patent Number: 7271192

Selective estrogen receptor-.beta. ligands
Inventor: Barlaam, et al. | Patent Number: 7256201

Aminobenzamide derivative
Inventor: Nishimura, et al. | Patent Number: 7253188

Benzisoxazolyl-, pyridoisoxazolyl-and benzthienyl-phenoxy derivatives useful as D.sub.4 antagonists
Inventor: Shutske, et al. | Patent Number: 7253165

Transfer hydrogenation process and catalyst
Inventor: Blacker, et al. | Patent Number: 7250526

Acetyl 2-hydroxy-1, 3-diaminoalkanes
Inventor: John, et al. | Patent Number: 7244725

Composition, process of making, and medical use of substituted 4-phenyltetrahydroisoquinolines
Inventor: Hofmeister, et al. | Patent Number: 7241775

Substituted tetrahydroisoquinoline compounds, methods of making, and their use
Inventor: Miller, et al. | Patent Number: 7241774

Nitrogen-containing compounds having kinase inhibitory activity and drugs containing the same
Inventor: Takami, et al. | Patent Number: 7217722

CCR5 modulators
Inventor: Armour, et al. | Patent Number: 7217714

Propanolamine derivatives
Inventor: Taniguchi, et al. | Patent Number: 7217706

Isoquinoline compounds
Inventor: Poissonnier-Durieux, et al. | Patent Number: 7214689

5-HT.sub.7 receptor antagonists
Inventor: Jover, et al. | Patent Number: 7211585

5-HT7 receptor ligands
Inventor: Jover, et al. | Patent Number: 7211584

N-[4-(heteroarylmethyl)phenyl]-heteroarylamines
Inventor: Venet, et al. | Patent Number: 7205312

Compounds useful for modulating abnormal cell proliferation
Inventor: Roifman, et al. | Patent Number: 7202383

Chemokine receptor binding heterocyclic compounds
Inventor: Bridger, et al. | Patent Number: 7183273

Process for the synthesis of derivatives of 2,3-dihydro-1,4-dioxino-[2,3-f] quinoline
Inventor: Chan, et al. | Patent Number: 7166723

Serine protease inhibitors
Inventor: Lively, et al. | Patent Number: 7157585

Benzene acetamide compounds useful as serine protease inhibitors
Inventor: Bisacchi, et al. | Patent Number: 7144895

Synthesis of enantiomerically pure amino-substituted fused bicyclic rings
Inventor: McEachern, et al. | Patent Number: 7135570

Preparation of fused polycyclic alkaloids by ring closure of azomethine ylides, novel compounds thereof and their use as chemotherapeutic agents
Inventor: Banwell, et al. | Patent Number: 7122673

Phenylglycine derivatives useful as serine protease inhibitors
Inventor: Glunz, et al. | Patent Number: 7122559

Cyclic diamines and derivatives as factor Xa inhibitors
Inventor: Qiao | Patent Number: 7115646

5-substituted isoquinoline derivatives
Inventor: Yamada, et al. | Patent Number: 7094789

Use of compounds for decreasing activity of hormone-sensitive lipase
Inventor: Ebdrup, et al. | Patent Number: 7067517

Bicyclic and tricyclic hetroaromatic compounds
Inventor: Yuan, et al. | Patent Number: 7053093

Amidoheterocycles as modulators of the melanocortin-4 receptor
Inventor: Chaturvedula, et al. | Patent Number: 7049323

Naphthalene derivatives
Inventor: Brain, et al. | Patent Number: 7045533

Substituted 3-aryl-5-aryl-[1,2,4]-oxadiazoles and analogs as activators of caspases and inducers of apoptosis and the use thereof
Inventor: Cai, et al. | Patent Number: 7041685

CCR5 modulators
Inventor: Armour, et al. | Patent Number: 7041667

Iron catalyzed cross coupling reactions of aromatic compounds
Inventor: Furstner, et al. | Patent Number: 7026478

Preparation of substituted aromatic compounds
Inventor: Meudt, et al. | Patent Number: 7022857

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