Patent Class: Organic Compounds -- Part Of The Class 532-570 Series (544/350)

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3, 4-dihydroquinoxalin-2(1H)-ones for use as stearoyl CoA desaturase inhibitors
Inventor: Chisholm, et al. | Patent Number: 8148376

Fused pyrazine compounds useful for the treatment of degenerative and inflammatory diseases
Inventor: Andrews, et al. | Patent Number: 8148369

Fused pyrazine compounds useful for the treatment of degenerative and inflammatory diseases
Inventor: Andrews, et al. | Patent Number: 8138193

Fused pyrazine compounds useful for the treatment of degenerative and inflammatory diseases
Inventor: Andrews, et al. | Patent Number: 8133895

Pyrido[2,3-B]pyrazine derivatives useful as herbicidal compounds
Inventor: Carter, et al. | Patent Number: 8133847

Imidazo[1,2-a]pyrazines as orexin receptor antagonists
Inventor: Alvaro, et al. | Patent Number: 8129384

Diketo substituted pyrrolo[2,3-C]pyridines
Inventor: Wang, et al. | Patent Number: 8124615

Substituted pyrrolo[2,3-b]pyrazines and methods for kinase modulation, and indications therefor
Inventor: Ibrahim, et al. | Patent Number: 8119637

Pyrrolopyrazine kinase inhibitors
Inventor: DuBois, et al. | Patent Number: 8119636

Substituted pyrrolo[2,3b]pyrazines and methods for treatment of raf protein kinase-mediated indications
Inventor: Ibrahim, et al. | Patent Number: 8110576

Derivatives of pyrrolo-pyrazines having a kinase inhibitory activity and their biological applications
Inventor: Meijer, et al. | Patent Number: 8106050

Substituted pyrrolo [1,2-a] pyrazines as calcium channel blockers
Inventor: Zhang, et al. | Patent Number: 8101614

6,6-bicyclic ring substituted heterobicyclic protein kinase inhibitors
Inventor: Arnold, et al. | Patent Number: 8101613

Process for the preparation of Sitagliptin
Inventor: Allegrini, et al. | Patent Number: 8097724

Pyrrolidine compounds
Inventor: Jiaang, et al. | Patent Number: 8071787

Eszopiclone process
Inventor: Mandava, et al. | Patent Number: 8058438

Compound having affinity to amyloid
Inventor: Tanifuji, et al. | Patent Number: 8022207

Substituted tetrahydropyrrolopyrazine compounds and the use thereof in the treatment and/or inhibition of pain
Inventor: Merla, et al. | Patent Number: 8017772

Substituted triazolopyrazines useful for the treatment of degenerative and inflammatory diseases
Inventor: Andrews, et al. | Patent Number: 8012983

Pyrrolopyrazinyl urea kinase inhibitors
Inventor: Bamberg, et al. | Patent Number: 8012974

Substituted indazoles as glucokinase activators
Inventor: Cao, et al. | Patent Number: 8008332

Pyrrolopyrazine kinase inhibitors
Inventor: Bamberg, et al. | Patent Number: 8008298

Phosphatidylinositol 3-kinase inhibitors and methods of their use
Inventor: Bajjalieh, et al. | Patent Number: 7989622

Method for producing substituted imidazo[1,2-A]pyrazines of (s)-1-(3-(2-sec-butyl-6-(1h-indol-3-yl)-3-oxo-3,7-dihydroimadazo[1,2-a]py- razin-8-yl)propyl)guanidine
Inventor: Ohmiya, et al. | Patent Number: 7989621

Indole derivatives and their use as medicament
Inventor: Emig, et al. | Patent Number: 7989453

Heteroaryl compounds, compositions thereof, and methods of treatment therewith
Inventor: Mortensen, et al. | Patent Number: 7981893

Multi-cyclic cinnamide derivatives
Inventor: Kimura, et al. | Patent Number: 7973033

Process for the resolution of zopiclone and intermediate compounds
Inventor: Bleda, et al. | Patent Number: 7968712

Diketo substituted pyrrolo[2,3-c] pyridines
Inventor: Wang, et al. | Patent Number: 7960406

Dipeptidyl peptidase inhibitors
Inventor: Feng, et al. | Patent Number: 7960384

Certain 1H-imidazo[4,5-B]pyrazin-2(3H)-ones and 1H-imidazo[4,5-B]pyrazin-2-ols, compositions thereof, and methods for their use
Inventor: Muci, et al. | Patent Number: 7956056

Substituted spirocyclic chromanamine compounds as Beta-Secretase modulators and methods of use
Inventor: La, et al. | Patent Number: 7951838

Folates, compositions and uses thereof
Inventor: Valoti, et al. | Patent Number: 7947662

Heterobicyclic compounds useful as kinase inhibitors
Inventor: Dhar, et al. | Patent Number: 7943617

Azaindoles for inhibiting aurora2 and other kinases
Inventor: Cox, et al. | Patent Number: 7943616

Thiazolopyridin-2-yloxy-phenyl and thiazolopyrazin-2-yloxy-phenyl amines as modulators of leukotriene A4 hydrolase
Inventor: Bacani, et al. | Patent Number: 7939527

Substituted biaryl quinolin-4-ylamine analogues
Inventor: Bakthavatchalam, et al. | Patent Number: 7935702

Pyrrolopyrazine kinase inhibitors
Inventor: DuBois, et al. | Patent Number: 7932254

Inhibitors of Akt activity
Inventor: Arruda, et al. | Patent Number: 7910561

Pyridine [3,4-b] pyrazinones
Inventor: Hughes, et al. | Patent Number: 7902195

5,6-di-substituted oxadiazolopyrazines and thiadiazolopyrazines as CXC-chemokine receptor ligands
Inventor: Biju | Patent Number: 7897606

Pyridol[2,3-B]pyrazinones for use as stearoyl CoA desaturase inhibitors
Inventor: Koltun, et al. | Patent Number: 7893066

Imidazolopyrazine compounds useful for the treatment of degenerative and inflammatory diseases
Inventor: Andrews, et al. | Patent Number: 7893058

Cyclohexyl or piperidinyl carboxamide antibiotic derivatives
Inventor: Hubschwerlen, et al. | Patent Number: 7888359

Aminopiperidines as dipeptidyl peptidase-IV inhibitors for the treatment or prevention of diabetes
Inventor: Cox, et al. | Patent Number: 7884104

Dipeptidyl Peptidase-IV inhibiting compounds, method of preparing the same, and pharmaceutical compositions containing the same as an active agent
Inventor: Lee, et al. | Patent Number: 7879848

Near-infrared-absorbing material and near-infrared-absorbing filter
Inventor: Kimura, et al. | Patent Number: 7875215

Process for the preparation of an optically active 5H-pyrrolo [3,4-B] pyrazine derivative
Inventor: Pillai, et al. | Patent Number: 7863273

IL-12 modulatory compounds
Inventor: Demko, et al. | Patent Number: 7863270

Bicyclic carbamoylpyridone derivative having HIV integrase inhibitory activity
Inventor: Yoshida, et al. | Patent Number: 7858788

Pyrrolo[1,2-a] pyrazin-1(2H)-one and pyrrolo[1,2-d][1,2,4]triazin-1(2H)-one derivatives as inhibitors of poly(ADP-ribose)polymerase (PARP)
Inventor: Jones, et al. | Patent Number: 7834015

Pharmaceutical compositions as inhibitors of dipeptidyl peptidase-IV (DPP-IV)
Inventor: Pei, et al. | Patent Number: 7834012

Inhibitors of bruton's tyrosine kinase
Inventor: Honigberg, et al. | Patent Number: 7825118

HIV integrase inhibitors
Inventor: Williams, et al. | Patent Number: 7820680

Tetrahydrotriazolopyrazine derivatives and uses thereof
Inventor: Harbeson | Patent Number: 7820666

Substitued [1,2,4]triazolo[1,5-a]pyrazines as dipeptidyl peptidase-IV inhibitors for the treatment or prevention of diabetes
Inventor: Biftu, et al. | Patent Number: 7812027

Substituted pyrano [2,3-b] pyridinamine compounds as beta-secretase modulators and methods of use
Inventor: Graceffa, et al. | Patent Number: 7803809

Pyrazole derivatives, compositions containing such compounds and methods of use
Inventor: Parmee, et al. | Patent Number: 7799818

Bicyclic piperazine compound having TGR23 antagonistic activity
Inventor: Fukatsu, et al. | Patent Number: 7795267

Pyrrolopyrazines and pyrazolopyrazines useful as inhibitors of protein kinases
Inventor: Binch, et al. | Patent Number: 7795259

Monocyclic and bicyclic compounds and methods of use
Inventor: Zhang, et al. | Patent Number: 7790726

Process for the preparation of eszopiclone
Inventor: Sawant, et al. | Patent Number: 7786304

Azaindazole compounds and methods of use
Inventor: Zhang, et al. | Patent Number: 7777035

Hexahydroimidazopyrazin-3-one compounds useful as modulators of androgen receptor function
Inventor: Balog, et al. | Patent Number: 7776859

Process for the resolution of zopiclone and intermediate compounds
Inventor: Bleda, et al. | Patent Number: 7772396

Piperazine-piperidines with CXCR3 antagonist activity
Inventor: Yu, et al. | Patent Number: 7763616

Substituted hexahydropyrazino [1,2-A] pyrimidine-4,7-dione derivatives, process for their preparation and their use as medicaments
Inventor: Flohr, et al. | Patent Number: 7750005

Triazolopyrazine derivatives
Inventor: Cheng, et al. | Patent Number: 7732604

Organic compounds as agents for the treatment of aldosterone mediated conditions
Inventor: Mc Kenna | Patent Number: 7732603

Inhibitors of Bruton's tyrosine kinase
Inventor: Verner | Patent Number: 7732454

Pyrido[2,3-B] pyrazin-3(4H)-ones for use as stearoyl CoA desaturase inhibitors
Inventor: Koltun, et al. | Patent Number: 7732453

Dipeptidyl peptidase inhibitors
Inventor: Gwaltney, et al. | Patent Number: 7732446

Non-nucleoside reverse transcriptase inhibitors
Inventor: Kennedy-Smith, et al. | Patent Number: 7713974

Imidazo based heterocycles
Inventor: Calderwood, et al. | Patent Number: 7709468

Indole derivatives as selective androgen receptor modulators (SARMS)
Inventor: Lanter, et al. | Patent Number: 7705147

Muscarinic agents as therapeutic compounds
Inventor: Buffat, et al. | Patent Number: 7691857

Triazolopyrazines and methods of making and using the same
Inventor: Dowling, et al. | Patent Number: 7674791

1-phenylalkanecarboxylic acid derivatives for the treatment of neurodegenerative diseases
Inventor: Raveglia, et al. | Patent Number: 7662995

Unsaturated mTOR inhibitors
Inventor: Crew, et al. | Patent Number: 7659274

Compounds for the treatment of inflammatory disorders
Inventor: Guo, et al. | Patent Number: 7652020

2-(R)-(4-fluoro-2-methyl-phenyl)-4-(S)-((8aS)-6-oxo-hexahydro-pyrrolo[1,2-- a]-pyrazin-2-yl)-piperidine-1-carboxylic acid [1-(R)-3,5-bis-trifluoromethyl-phenyl)-ethyl]-methylamide maleate and pharmaceutical compositions thereof
Inventor: Alvaro, et al. | Patent Number: 7652012

Nitrogen-substituted hexahydropyrazino[1,2-A]pyrimidine-4,7-dione derivatives, processes for their preparation and their use as medicaments
Inventor: Flohr, et al. | Patent Number: 7652007

Bicyclic protein kinase inhibitors
Inventor: Crew, et al. | Patent Number: 7648987

Phenyl-aniline substituted bicyclic compounds useful as kinase inhibitors
Inventor: Das, et al. | Patent Number: 7642257

Compounds for the treatment of inflammatory disorders
Inventor: Siddiqui, et al. | Patent Number: 7638513

Method for producing .beta.-heteroaryl-.alpha.-alanine compounds using 2-amino-2-(heteroarylmethyl) carboxylic acid compounds
Inventor: Oehlinger | Patent Number: 7626022

Fused ring heterocycle kinase modulators
Inventor: Arnold, et al. | Patent Number: 7626021

Intermediate compounds for the manufacture of fused piperazin-2-one derivatives
Inventor: Duran, et al. | Patent Number: 7626019

Substituted monocyclic CGRP receptor antagonists
Inventor: Wood, et al. | Patent Number: 7625901

Sutstituted tetrahydropyrrolopyrazine compounds and the use thereof in the treatment and/or inhibition of pain
Inventor: Merla, et al. | Patent Number: 7625900

Pyridodihydropyraziones, process for their manufacture and use thereof as medicaments
Inventor: Hoffmann, et al. | Patent Number: 7625899

Amorphous form of a phosphoric acid salt of a dipeptidyl peptidase-IV inhibitor
Inventor: Ferlita, et al. | Patent Number: 7612072

Indole derivative having heterocycle and mono- or diazaindole derivative
Inventor: Matsuoka, et al. | Patent Number: 7612070

Imidazo[4,5-b]pyrazinone inhibitors of protein kinases
Inventor: Liu, et al. | Patent Number: 7608622

Substituted pyrazolo[3,4-d]pyrimidines as p38 MAP kinase inhibitors
Inventor: Arora, et al. | Patent Number: 7601726

Pyridopyrazines and derivatives thereof as ALK and c-Met inhibitors
Inventor: Dorsey, et al. | Patent Number: 7601716

Quinoxaline derivative, and organic semiconductor device, electric field light emitting device, and electronic device which have the same
Inventor: Shitagaki, et al. | Patent Number: 7601435

Certain 1H-imidazo[4,5-b]pyrazin-2(3H)-ones and 1H-imidazo[4,5-b]pyrazin-2-ols, compositions thereof, and methods for their use
Inventor: Muci, et al. | Patent Number: 7598248

Inhibitors of Akt activity
Inventor: Cosford, et al. | Patent Number: 7589068

Reverse-turn mimetics and method relating thereto
Inventor: Moon, et al. | Patent Number: 7585862

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