Patent Class: Organic Compounds -- Part Of The Class 532-570 Series (544/328)

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Substituted pyrimidinyl oxime kinase inhibitors
Inventor: Xu, et al. | Patent Number: 8153791

Pyrimidine derivatives which are antagonist of the vitronectin receptor
Inventor: Lefrancois, et al. | Patent Number: 8133896

Pyrimidine compound and pests controlling composition containing the same
Inventor: Mizuno, et al. | Patent Number: 8129526

Process for the synthesis of 5-(methyl-1H-imidazol-1-yl)-3-(trifluoromethyl)-benzeneamine
Inventor: Shieh, et al. | Patent Number: 8124763

Fungicide hydroximoyl-tetrazole derivatives
Inventor: Christian, et al. | Patent Number: 8119646

Fungicide hydroximoyl-tetrazole derivatives
Inventor: Christian, et al. | Patent Number: 8119645

(1H-indol-7-yl)-(pyrimidin-2-ylamino)methanone derivatives and related compounds as IGF-R1 inhibitors for the treatment of cancer
Inventor: Heinrich, et al. | Patent Number: 8114882

Aminopyridine derivatives having aurora a selective inhibitory action
Inventor: Kato, et al. | Patent Number: 8101621

Cyanopyrimidinones
Inventor: Hendrix, et al. | Patent Number: 8088769

Benzimidazoles useful as inhibitors of protein kinases
Inventor: Binch, et al. | Patent Number: 8076343

Polymorphs of dasatinib isopropyl alcohol and process for preparation thereof
Inventor: {hacek over (S)}imo, et al. | Patent Number: 8067423

Substituted dihydropyrazolones and their use
Inventor: Jeske, et al. | Patent Number: 8067407

N-heterocyclic inhibitors of TNF-alpha expression
Inventor: Ahmed, et al. | Patent Number: 8044040

Calcium channel antagonists
Inventor: Pacofsky, et al. | Patent Number: 8034954

[4,5']Bipyrimidinyl-6,4'-diamine derivatives as protein kinase inhibitors
Inventor: Albaugh, et al. | Patent Number: 8026243

Aurora kinase modulators and method of use
Inventor: Cee, et al. | Patent Number: 8022221

Pyrazole compounds useful as protein kinase inhibitors
Inventor: Bebbington, et al. | Patent Number: 7982037

Anhydrous form of dasatinib and process for preparation thereof
Inventor: {hacek over (S)}imo, et al. | Patent Number: 7973045

Pyrimidine compound and pests controlling composition containing the same
Inventor: Mizuno, et al. | Patent Number: 7928110

6-substituted 2-(benzimidazolyl)purine and purinone derivatives for immunosuppression
Inventor: Neagu, et al. | Patent Number: 7919490

Substituted heterocycles and methods of use
Inventor: Bellon, et al. | Patent Number: 7915287

8-substituted 2-(benzimidazolyl)purine derivatives for immunosuppression
Inventor: Lu, et al. | Patent Number: 7915268

6-substituted 2-(benzimidazolyl)purine and purinone derivatives for immunosuppression
Inventor: Neagu, et al. | Patent Number: 7902187

Hydrazone derivatives as kinase inhibitors
Inventor: Xu, et al. | Patent Number: 7893064

Tyrosine kinase inhibitors containing a zinc binding moiety
Inventor: Cai, et al. | Patent Number: 7888361

Aminopiperidines as dipeptidyl peptidase-IV inhibitors for the treatment or prevention of diabetes
Inventor: Cox, et al. | Patent Number: 7884104

4,6-disubstituted pyrimidines and their use as protein kinase inhibitors
Inventor: Stadlwieser, et al. | Patent Number: 7879853

Compositions useful as inhibitors of GSK-3
Inventor: Forster, et al. | Patent Number: 7872129

Heterocycles
Inventor: Srinivas, et al. | Patent Number: 7863446

Heteromonocyclic compound or a salt thereof having strong antihypertensive action, insulin sensitizing activity and the like production thereof and use thereof for prophylaxis or treatment of cardiovascular diseases, metabolic diseases and/or central nervous system diseases
Inventor: Kuroita, et al. | Patent Number: 7803940

Substituted 3-carboxamido isoxazoles as kinase modulators
Inventor: Mehta, et al. | Patent Number: 7767670

Pyrimidine carboxamides
Inventor: Tadipartiii, et al. | Patent Number: 7759350

Therapeutic agents useful for treating pain
Inventor: Sun, et al. | Patent Number: 7754723

Compounds and compositions as protein kinase inhibitors
Inventor: Ren, et al. | Patent Number: 7745437

Compounds and compositions useful as cathepsin S inhibitors
Inventor: Hart, et al. | Patent Number: 7704996

Therapeutic agents useful for treating pain
Inventor: Kyle, et al. | Patent Number: 7683063

Pyrimidine derivatives for treatment of hyperproliferative disorders
Inventor: Dixon, et al. | Patent Number: 7678804

Substituted biaryl piperazinyl-pyridine analogues
Inventor: Blum, et al. | Patent Number: 7662830

Pteridinone derivatives for use as stearoyl CoA desaturase inhibitors
Inventor: Chisholm, et al. | Patent Number: 7662819

Urea or thiourea substituted 1,4-pyrazine compounds useful as anti-cancer agents and for inhibiting Chk1
Inventor: Kesicki, et al. | Patent Number: 7608618

Pyrimidine derivatives for treatment of hyperproliferative disorders
Inventor: Dixon, et al. | Patent Number: 7582645

Met kinase inhibitors
Inventor: Borzilleri, et al. | Patent Number: 7547782

Compounds which inhibit leukocyte adhesion mediated by VLA-4
Inventor: Konradi, et al. | Patent Number: 7538215

Vanilloid receptor ligands and their use in treatments
Inventor: Balan, et al. | Patent Number: 7534798

5-arylpyrimidines as anticancer agents
Inventor: Zhang, et al. | Patent Number: 7524849

Heteroaryl amines as glycogen synthase kinase 3.beta. inhibitors (GSK3 inhibitors)
Inventor: Freyne, et al. | Patent Number: 7514445

11b-HSD1 inhibitors for the treatment of diabetes
Inventor: Amrein, et al. | Patent Number: 7507733

Compositions useful as inhibitors of GSK-3
Inventor: Forster, et al. | Patent Number: 7491730

Pyrazole compounds useful as protein kinase inhibitors
Inventor: Davies, et al. | Patent Number: 7473691

Pyridine derivatives as Raf kinase inhibitors
Inventor: Bamford, et al. | Patent Number: 7452906

Triazole compounds useful in therapy
Inventor: Bryans, et al. | Patent Number: 7442795

Purine-or pyrrolol[2,3-d]pyrimidine-2-carbonitiles for treating diseases associated with cysteine protease activity
Inventor: Bailey, et al. | Patent Number: 7439240

Utilities of amide compounds
Inventor: Yamamori, et al. | Patent Number: 7429593

Pyrimidines and uses thereof
Inventor: Bhatt, et al. | Patent Number: 7419984

Pyridine-2-carboxyamide derivatives
Inventor: Jaeschke, et al. | Patent Number: 7414060

Pyrazolyl and imidazolyl pyrimidines as CRF antagonists
Inventor: Jahangir, et al. | Patent Number: 7414059

4-amino-substituted pyrimidine derivatives
Inventor: Feurer, et al. | Patent Number: 7410973

Pyrazole compounds useful as protein kinase inhibitors
Inventor: Davies, et al. | Patent Number: 7390815

Phosphodiesterase 4 inhibitors
Inventor: Hopper, et al. | Patent Number: 7335654

2-(2-pyridyl)-5-phenyl-6-aminopyrimidine, method and intermediate products for the production and use thereof for combating noxious fungi
Inventor: Schieweck, et al. | Patent Number: 7320975

Methods of treating medical conditions using sulfonate-substituted pyrazolopyridine derivatives
Inventor: Stasch, et al. | Patent Number: 7317016

Heteroaryl urea neuropeptide Y Y5 receptor antagonists
Inventor: Stamford, et al. | Patent Number: 7309704

Chemical compounds
Inventor: Hiscock, et al. | Patent Number: 7294627

Medical uses of carbamate-substituted pyrazolo-pyridine derivatives
Inventor: Stasch, et al. | Patent Number: 7291622

N-heterocyclic inhibitors of TNF-.alpha. expression
Inventor: Ahmed, et al. | Patent Number: 7253174

Substituted 2-aryl-4-arylaminopyrimidines and analogs as activators of caspases and inducers of apoptosis and the use thereof
Inventor: Cai, et al. | Patent Number: 7226927

Substituted pyrazinones, pyridines and pyrimidines as corticotropin releasing factor ligands
Inventor: Arvanitis, et al. | Patent Number: 7205306

Methods and compositions as protein kinase inhibitors
Inventor: Chopiuk, et al. | Patent Number: 7189729

Carbamate-substituted pyrazolopyridines
Inventor: Alonso-Alija, et al. | Patent Number: 7173037

Aminopyrimidine and aminopyridine anti-inflammation agents
Inventor: Hawley, et al. | Patent Number: 7157580

5-Phenylpyrimidines, methods and intermediate products for the production thereof and use of the same for controlling pathogenic fungi
Inventor: Grote, et al. | Patent Number: 7153860

Derivatives of 2-(1-benzyl-1H-pyrazolo(3,4-B)pyridine-3-yl)-5(-4-pyridinyl)l-4-pyrimidin- amines and the use thereof as quanylate cyclase stimulators
Inventor: Weigand, et al. | Patent Number: 7135474

Sulfonamide-substituted pyrazolopyridine compounds
Inventor: Stasch, et al. | Patent Number: 7115599

Tyrosine kinase inhibitors
Inventor: Bilodeau, et al. | Patent Number: 7115597

Cysteine protease inhibitors with 2-cyano-4-amino-pyrimidine structure and cathepsin k inhibitory activity for the treatment of inflammations and other diseases
Inventor: Altmann, et al. | Patent Number: 7112589

Carbamate-substituted pyrazolopyridine-derivatives
Inventor: Stasch, et al. | Patent Number: 7105523

Compositions useful as inhibitors of protein kinases
Inventor: Bebbington, et al. | Patent Number: 7091343

2,5-disubstituted pyrimidine derivatives
Inventor: Feurer, et al. | Patent Number: 7091198

Pyrazolyl pyrimidines
Inventor: Fischer, et al. | Patent Number: 7087616

2,4,DI (hetero-) arylamino (-oxy)-5-substituted pyrimidines as antineoplastic agents
Inventor: Pease, et al. | Patent Number: 7067522

N-substituted nonaryl-heterocyclic NMDA/NR2B antagonists
Inventor: Claiborne, et al. | Patent Number: 7053089

Modulators of TNF-.alpha. signaling
Inventor: Sneddon, et al. | Patent Number: 7034031

Prodrugs of HIV replication inhibiting pyrimidines
Inventor: Kukla, et al. | Patent Number: 7034019

4-amino-2-(2-pyridyl)pyrimidines as microbicidal active substances
Inventor: Haap, et al. | Patent Number: 7015228

Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by VLA-4
Inventor: Konradi, et al. | Patent Number: 7005433

Beta-amino acid derivatives-inhibitors of leukocyte adhesion mediated by VLA-4
Inventor: Konradi, et al. | Patent Number: 6953802

Bradykinin B1 receptor antagonists
Inventor: Ohlmeyer, et al. | Patent Number: 6919347

Sulfonate substituted pyrazol pyridine derivatives
Inventor: Stasch, et al. | Patent Number: 6919345

Lactam-substituted pyrazolopyridine derivatives
Inventor: Stasch, et al. | Patent Number: 6903089

Heterocyclic sodium/proton exchange inhibitors and method
Inventor: Ahmad, et al. | Patent Number: 6887870

6-(1-fluoroethyl)-5-iodo-4-aminopyrimidine compounds process for preparation of the same and pest controllers for agricultural and horticultural use
Inventor: Fujii, et al. | Patent Number: 6867212

Pyridine and pyrimidine derivatives
Inventor: Boehringer, et al. | Patent Number: 6867205

N-heterocyclic derivatives as NOS inhibitors
Inventor: Arnaiz, et al. | Patent Number: 6864263

Pyrimidine compounds
Inventor: Sun, et al. | Patent Number: 6858606

N-heterocyclic derivatives as NOS inhibitors
Inventor: Arnaiz, et al. | Patent Number: 6846829

Aminopyrimidine and aminopyridine anti-inflammation agents
Inventor: Hawley, et al. | Patent Number: 6846828

Pyrimidine derivatives
Inventor: Cumming | Patent Number: 6846827

N-heterocyclic derivatives as NOS inhibitors
Inventor: Arnaiz, et al. | Patent Number: 6841674

2,4-Di(hetero-)arylamino(-oxy)-5-substituted pyrimidines as antineaoplastic agents
Inventor: Pease, et al. | Patent Number: 6838464

Substituted pyrazole derivatives
Inventor: Straub, et al. | Patent Number: 6833364

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