Patent Class: Drug, Bio-Affecting And Body Treating Compositions (514/326)

Description

Class 514 is an integral part of Class 424. It incorporatesall the definitions and rules as to subject matter of Class 424.

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Quaternary ammonium salts as M3 antagonists
Inventor: Press, et al. | Patent Number: 8153669

Piperidine derivative or salt thereof
Inventor: Hachiya, et al. | Patent Number: 8153658

Dopamine-, norepinephrine- and serotonin-transporter-selective heterocyclic compounds and their therapeutic applications
Inventor: Kozikowski, et al. | Patent Number: 8153657

Modulators of CB1 receptors
Inventor: Cooper, et al. | Patent Number: 8148404

Thrombopoietin mimetics
Inventor: Spencer, et al. | Patent Number: 8143287

Piperidine derivative
Inventor: Ishikawa, et al. | Patent Number: 8138206

Isoxazole derivatives and pharmaceutical compositions comprising the same
Inventor: Tzeng, et al. | Patent Number: 8138184

Biphenyl compounds useful as muscarinic receptor antagonists
Inventor: Mu, et al. | Patent Number: 8133905

Dihydroindolone compounds, a process for their preparation and pharmaceutical compositions containing them
Inventor: Ortuno, et al. | Patent Number: 8133889

Crystalline forms of MC4R agonist and process for synthesis
Inventor: Calabria, et al. | Patent Number: 8129413

Hydantoin derivatives useful as metalloproteinase inhibitors
Inventor: Waterson, et al. | Patent Number: 8129412

Substituted pyrazole and triazole compounds as KSP inhibitors
Inventor: Xia, et al. | Patent Number: 8129358

Biphenyl compounds useful as muscarinic receptor antagonists
Inventor: Mu, et al. | Patent Number: 8124627

Substituted sulfonamide compounds
Inventor: Oberboersch, et al. | Patent Number: 8124624

Pharmaceutical compositions as inhibitors of dipeptidyl peptidase-IV (DPP-IV)
Inventor: Madar, et al. | Patent Number: 8119664

Heteroaryl-substituted piperidines
Inventor: Heimbach, et al. | Patent Number: 8119663

Derivatives of 4-aminopiperidine and their use as a medicament
Inventor: Thurieau, et al. | Patent Number: 8110574

Benzoyl-piperidine derivatives as dual modulators of the 5-HT2A and D3 receptors
Inventor: Gobbi, et al. | Patent Number: 8097637

Pharmaceutical compositions comprising 2-methoxy-5-(5-trifluoromethyl-tetrazol-1-yl-benzyl)-(2S-phenylpiperidin-- 3S-yl-)
Inventor: Alvaro, et al. | Patent Number: 8093268

Nitrogen-containing heterocyclic compounds and thrombopoietin receptor activators
Inventor: Miyaji, et al. | Patent Number: 8093251

Cannabinoid receptor antagonists/inverse agonists useful for treating obesity
Inventor: McElroy, et al. | Patent Number: 8088798

Substituted N-(4-cyano-1H-pyrazol-3-yl)methylamine derivatives, preparation thereof and therapeutic use thereof
Inventor: Barth, et al. | Patent Number: 8088797

Biphenyl amide lactam derivatives as inhibitors of 11-beta-hydroxysteroid dehydrogenase 1
Inventor: Aicher, et al. | Patent Number: 8088776

Substituted piperidines
Inventor: Heimbach, et al. | Patent Number: 8084469

Pyrazole derivatives as cannabinoid receptor antagonists
Inventor: Makriyannis, et al. | Patent Number: 8084467

Organic compounds
Inventor: Neubert, et al. | Patent Number: 8084448

Biphenyl compounds useful as muscarinic receptor antagonists
Inventor: Mammen, et al. | Patent Number: 8067439

Nitric oxide enhancing prostaglandin compounds, compositions and methods of use
Inventor: Garvey | Patent Number: 8067414

Oxadiazole derivatives and thiadiazole derivatives having neovascularization inhibitory activity
Inventor: Honda, et al. | Patent Number: 8063034

Diacylglycerol acyltransferase inhibitors
Inventor: Bolin, et al. | Patent Number: 8058299

3-imidazolyl-indoles for the treatment of proliferative diseases
Inventor: Boettcher, et al. | Patent Number: 8053457

Pyrrole derivatives, preparation thereof and therapeutic use thereof
Inventor: Barth, et al. | Patent Number: 8044072

Method for reducing side effects of CB.sub.2 receptor agonist therapy using a combination of a selective CB.sub.2 receptor agonist and a selective CB.sub.1 receptor antagonist
Inventor: Carroll | Patent Number: 8044071

Sulfonamide substituted pyrazoline compounds, their preparation and use as CB1 modulators
Inventor: Buschmann, et al. | Patent Number: 8044053

Benzoyl-piperidine derivatives as dual modulators of the 5-HT2A and D3 receptors
Inventor: Gobbi, et al. | Patent Number: 8039490

Guanidine-containing compounds useful as muscarinic receptor antagonists
Inventor: Ji, et al. | Patent Number: 8039489

Piperidine-amide derivatives
Inventor: Andjelkovic, et al. | Patent Number: 8039487

Allosteric modulators of metabotropic glutamate receptors
Inventor: Bessis, et al. | Patent Number: 8030331

Therapeutic agents useful for treating pain
Inventor: Chen | Patent Number: 8026254

Pyrrole derivatives as pharmaceutical agents
Inventor: Canne Bannen, et al. | Patent Number: 8026237

Pyrrolidine derivatives
Inventor: Jiaang, et al. | Patent Number: 8022096

5-Phenylthiazole derivatives and their use as p13 kinase inhibitors
Inventor: Bloomfield, et al. | Patent Number: 8017608

N-substituted-pyrrolidines as inhibitors of MDM2-P-53 interactions
Inventor: Bartkovitz, et al. | Patent Number: 8017607

Pharmaceutically active sulfonamide derivatives
Inventor: Arkinstall, et al. | Patent Number: 8012995

N-hydroxyamide derivatives and use thereof
Inventor: Swinnen, et al. | Patent Number: 8008302

Histamine H3 receptor agents, preparation and therapeutic uses
Inventor: Beavers, et al. | Patent Number: 8008296

Hydantoin derivatives useful as antibacterial agents
Inventor: Mansoor, et al. | Patent Number: 7998961

Therapeutic substituted piperidone compounds
Inventor: Old, et al. | Patent Number: 7994195

Imidazole compounds having pharmaceutical activity towards the sigma receptor
Inventor: Cuberes-Altisent, et al. | Patent Number: 7989485

Substituted pyrazoles, compositions containing such compounds and methods of use
Inventor: Parmee, et al. | Patent Number: 7989475

1,5 and 3,6-substituted indole compounds having NOS inhibitory activity
Inventor: Maddaford, et al. | Patent Number: 7989447

1-oxyalkyl-2-carboxyl-7-nonsubstituted indole derivatives
Inventor: Song, et al. | Patent Number: 7981888

Prodrugs of ion channel modulating compounds and uses thereof
Inventor: Choi, et al. | Patent Number: 7977373

Pyrrole derivative having ureido group and aminocarbonyl group as substituents
Inventor: Kawashima, et al. | Patent Number: 7977371

Pyrazol derivatives
Inventor: Aebi, et al. | Patent Number: 7977358

1,3-disubstituted 4-methyl-1H-pyrrole-2-carboxamides and their use in medicaments
Inventor: Oberboersch, et al. | Patent Number: 7968591

Substituted N-aryl heterocycles, process for their preparation and their use as medicaments
Inventor: Schwink, et al. | Patent Number: 7968550

Non-anilinic derivatives of isothiazol-3(2H)-one 1,1-dioxides as liver X receptor modulators
Inventor: Broo, et al. | Patent Number: 7960380

Piperidines as chemokine modulators (CCR)
Inventor: Alcaraz, et al. | Patent Number: 7956070

Piperidinium and pyrrolidinium derivatives as ligands for the muscarinic M3 receptor
Inventor: Collingwood, et al. | Patent Number: 7947730

Substituted 5-vinylphenyl-1-phenyl-pyrazole cannabinoid modulators
Inventor: Xia, et al. | Patent Number: 7943653

Compounds comprising a lactam or a lactam derivative moiety, processes for making them, and their uses
Inventor: Celanire, et al. | Patent Number: 7943605

Compounds and compositions as channel activating protease inhibitors
Inventor: Tully, et al. | Patent Number: 7939547

Imidazole derivatives
Inventor: Aebi, et al. | Patent Number: 7935707

Use of .alpha.-glucosidase inhibitors to treat alphavirus infections
Inventor: Blatt, et al. | Patent Number: 7932267

Compounds which modulate the CB2 receptor
Inventor: Berry, et al. | Patent Number: 7928123

4-ethynyl pyrazole derivative compounds and methods for treatment of HCV
Inventor: Li, et al. | Patent Number: 7923004

Ubiquitin ligase inhibitors
Inventor: Ramesh, et al. | Patent Number: 7915293

1,3-oxazolidin-2-one derivatives useful as CETP inhibitors
Inventor: Ali, et al. | Patent Number: 7915271

Pyrazole-derivatives as factor Xa inhibitors
Inventor: Nazare, et al. | Patent Number: 7910606

Carbonyl compounds
Inventor: Tsaklakidis, et al. | Patent Number: 7906516

Diaminotriazoles useful as inhibitors of protein kinases
Inventor: Pierce, et al. | Patent Number: 7902239

Compounds 010
Inventor: Furber, et al. | Patent Number: 7902181

Pyrazoles for the treatment of obesity and other CNS disorders
Inventor: Bennani, et al. | Patent Number: 7897634

Substituted pyrazoline compounds, their preparation and use as medicaments
Inventor: Torrens, et al. | Patent Number: 7897589

Organic compounds
Inventor: Baeschlin, et al. | Patent Number: 7888351

Substituted piperidine compounds and methods of their use
Inventor: Dolle, et al. | Patent Number: 7884102

Thiazole derivatives and use thereof
Inventor: Quattropani, et al. | Patent Number: 7879888

Izoxazoline derivative and herbicide
Inventor: Nakatani, et al. | Patent Number: 7875606

Low molecular weight Myc-max inhibitors
Inventor: Metallo, et al. | Patent Number: 7872027

Ligand activators of the RAR receptors and pharmaceutical/cosmetic applications thereof
Inventor: Biadatti, et al. | Patent Number: 7872026

Substituted thiazoles and their use for producing drugs
Inventor: Haurand, et al. | Patent Number: 7871999

Substituted imidazole 4-carboxamides as cholecystokinin-1 receptor modulators
Inventor: Berger, et al. | Patent Number: 7858629

Piperidine and morpholine renin inhibitors
Inventor: Baldwin, et al. | Patent Number: 7858624

Compounds
Inventor: Alvaro, et al. | Patent Number: 7855218

Piperdine-based inhibitors of sodium glucose co-transporter 2 and methods of their use
Inventor: Harrison, et al. | Patent Number: 7846945

Nicotine receptor agonists in stem cell and progenitor cell recruitment
Inventor: Cooke, et al. | Patent Number: 7838539

Substituted pyrazolyl urea derivatives useful in the treatment of cancer
Inventor: Lee, et al. | Patent Number: 7838524

Thiophene compounds
Inventor: Shia, et al. | Patent Number: 7834046

Allosteric modulators of metabotropic glutamate receptors
Inventor: Bessis, et al. | Patent Number: 7834035

Phenyl-[1,2,4]-oxadiazol-5-one derivatives, pharmaceutical compositions and therapeutic use thereof
Inventor: Keil, et al. | Patent Number: 7834030

5-aminopyrazole derivatives as pesticidal compounds
Inventor: Schnatterer, et al. | Patent Number: 7834003

CGRP receptor antagonists
Inventor: Gutierrez, et al. | Patent Number: 7834000

Prodrugs of pyrazoline compounds, their preparation and use as medicaments
Inventor: Torrens Jover, et al. | Patent Number: 7829581

Cyclic amine derivative having heteroaryl ring
Inventor: Kimura, et al. | Patent Number: 7829580

3,4-disubstituted 1H-pyrazole compounds and their use as cyclin dependent kinase and glycogen synthase kinase-3 modulators
Inventor: Berdini, et al. | Patent Number: 7825140

Compounds and methods for selective inhibition of dipeptidyl peptidase-IV
Inventor: Campbell, et al. | Patent Number: 7825139

Cyclized derivatives as Eg-5 inhibitors
Inventor: Boyce, et al. | Patent Number: 7820646

Tubulysin analogues
Inventor: Domling, et al. | Patent Number: 7816377

Ligands for monoamine receptors and transporters, and methods of use thereof
Inventor: Aquila, et al. | Patent Number: 7816375

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